Use and specificity of staurosporine, UCN-01, and calphostin C as protein kinase inhibitors

Methods Enzymol. 1991:201:340-7. doi: 10.1016/0076-6879(91)01030-6.
No abstract available

Publication types

  • Comparative Study

MeSH terms

  • Alkaloids / pharmacology*
  • Animals
  • Avian Sarcoma Viruses / genetics
  • Brain / enzymology
  • Cattle
  • Cell Line
  • Chick Embryo
  • Molecular Structure
  • Myocardium / enzymology
  • Naphthalenes*
  • Oncogene Protein pp60(v-src) / antagonists & inhibitors*
  • Polycyclic Compounds / pharmacology*
  • Protein Kinase C / antagonists & inhibitors*
  • Protein Kinase C / isolation & purification
  • Protein Kinase Inhibitors*
  • Protein Kinases / isolation & purification
  • Protein-Tyrosine Kinases / antagonists & inhibitors*
  • Protein-Tyrosine Kinases / isolation & purification
  • Rats
  • Staurosporine
  • Structure-Activity Relationship

Substances

  • Alkaloids
  • Naphthalenes
  • Polycyclic Compounds
  • Protein Kinase Inhibitors
  • 7-hydroxystaurosporine
  • Protein Kinases
  • Protein-Tyrosine Kinases
  • Oncogene Protein pp60(v-src)
  • Protein Kinase C
  • Staurosporine
  • calphostin C