Beta-adrenergic activities of octopamine and synephrine stereoisomers on guinea-pig atria and trachea

J Pharm Pharmacol. 1987 Sep;39(9):752-4. doi: 10.1111/j.2042-7158.1987.tb06986.x.

Abstract

The activities of the (-)- and (+)-forms of m- and p-octopamine and m- and p-synephrine on beta 1- and beta 2-adrenoceptors in guinea-pig atria and trachea have been compared with that of noradrenaline. The rank order of potency of the (-)-forms on beta 1-adrenoceptors was noradrenaline greater than m-synephrine greater than m-octopamine = p-octopamine greater than p-synephrine. m-Synephrine was 100-fold, m- and p-octopamine about 6000-fold, and p-synephrine about 40,000-fold less active than noradrenaline. The (+)-forms were 1-2 orders of magnitude less active than their (-)-counterparts. The four (-)-compounds were more than four orders of magnitude less active than noradrenaline on beta 2-adrenoceptors, and the (+)-forms had no detectable activity in concentrations as high as 10(-4) M. If m- and p-octopamine are co-released with noradrenaline in amounts proportional to their concentration, their activities at these structures are too low to be physiologically significant.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adrenergic beta-Agonists
  • Adrenergic beta-Antagonists
  • Animals
  • Guinea Pigs
  • Heart / drug effects*
  • In Vitro Techniques
  • Male
  • Muscle, Smooth / drug effects*
  • Octopamine / pharmacology*
  • Receptors, Adrenergic, beta / drug effects*
  • Stereoisomerism
  • Synephrine / pharmacology*
  • Trachea / drug effects

Substances

  • Adrenergic beta-Agonists
  • Adrenergic beta-Antagonists
  • Receptors, Adrenergic, beta
  • Octopamine
  • Synephrine