Circ_ZNF512-Mediated miR-181d-5p Inhibition Limits Cardiomyocyte Autophagy and Promotes Myocardial Ischemia/Reperfusion Injury through an EGR1/mTORC1/TFEB-Based Mechanism

J Med Chem. 2022 Feb 10;65(3):1808-1821. doi: 10.1021/acs.jmedchem.1c00745. Epub 2022 Jan 18.

Abstract

Studies have shown that circRNAs are important regulatory molecules involved in cell physiology and pathology. Herein, we analyzed the role of circ_ZNF512 in cardiomyocyte autophagy of myocardial ischemia/reperfusion (I/R) injury. A mouse model was induced by ligation of the left anterior descending artery followed by reperfusion. An in vitro model was also developed in cultured cardiomyocytes following hypoxia/reoxygenation (H/R) injury. It was established that EGR1 expression was increased in myocardial tissues of I/R mice and H/R-induced cardiomyocytes. Silencing of circ_ZNF512 attenuated its binding to miR-181d-5p, which in turn impaired the EGR1 expression by targeting its 3'-UTR, thus promoting the autophagy of cardiomyocytes and suppressing cell apoptosis to alleviate myocardial tissue injury. Additionally, the circ_ZNF512/miR-181d-5p/EGR1 crosstalk activated the mTORC1/TFEB signaling pathway, increasing mTORC1 expression while suppressing TFEB expression. Together, circ_ZNF512 knockdown protects against myocardial I/R injury, which may be a potential therapeutic approach for preventing myocardial I/R injury.

MeSH terms

  • Animals
  • Autophagy / physiology*
  • Basic Helix-Loop-Helix Leucine Zipper Transcription Factors / metabolism
  • Early Growth Response Protein 1 / metabolism
  • Male
  • Mechanistic Target of Rapamycin Complex 1 / metabolism
  • Mice
  • Mice, Inbred C57BL
  • MicroRNAs / metabolism*
  • Myocardial Reperfusion Injury / metabolism*
  • Myocytes, Cardiac / metabolism*
  • RNA, Circular / metabolism*
  • Signal Transduction / physiology

Substances

  • Basic Helix-Loop-Helix Leucine Zipper Transcription Factors
  • Early Growth Response Protein 1
  • Egr1 protein, mouse
  • MicroRNAs
  • RNA, Circular
  • Tcfeb protein, mouse
  • mirn181 microRNA, mouse
  • Mechanistic Target of Rapamycin Complex 1