Carazolol, an extremely potent beta-adrenergic blocker: binding to beta-receptors in brain membranes

Life Sci. 1979 Jun 11;24(24):2255-64. doi: 10.1016/0024-3205(79)90102-4.
No abstract available

MeSH terms

  • Adrenergic beta-Antagonists / blood
  • Adrenergic beta-Antagonists / metabolism*
  • Animals
  • Blood Proteins / metabolism
  • Brain / metabolism*
  • Carbazoles / blood
  • Carbazoles / metabolism*
  • Dihydroalprenolol / metabolism
  • Kinetics
  • Male
  • Membranes / metabolism
  • Propanolamines / blood
  • Propanolamines / metabolism*
  • Protein Binding
  • Rats
  • Receptors, Adrenergic / metabolism*
  • Receptors, Adrenergic, beta / metabolism*

Substances

  • Adrenergic beta-Antagonists
  • Blood Proteins
  • Carbazoles
  • Propanolamines
  • Receptors, Adrenergic
  • Receptors, Adrenergic, beta
  • carazolol
  • Dihydroalprenolol