Accumulation of cyclic adenosine monophosphate in incubated slices of brain tissue. 1. Structure-activity relationships of agonists and antagonists of biogenic amines and of tricyclic tranquilizers and antidepressants

J Med Chem. 1972 May;15(5):458-62. doi: 10.1021/jm00275a004.
No abstract available

MeSH terms

  • Adrenergic alpha-Antagonists / pharmacology
  • Adrenergic beta-Antagonists / pharmacology
  • Animals
  • Antidepressive Agents / pharmacology*
  • Brain / metabolism*
  • Brain Chemistry / drug effects
  • Carbon Isotopes
  • Catecholamines / pharmacology*
  • Cerebral Cortex / metabolism
  • Cyclic AMP / metabolism*
  • Epinephrine / pharmacology
  • Guinea Pigs
  • Hallucinogens / pharmacology
  • Histamine / pharmacology*
  • Histamine H1 Antagonists / pharmacology
  • In Vitro Techniques
  • Isoproterenol / pharmacology
  • Monoamine Oxidase Inhibitors / pharmacology
  • Norepinephrine / pharmacology
  • Serotonin / pharmacology*
  • Structure-Activity Relationship
  • Tranquilizing Agents / pharmacology*

Substances

  • Adrenergic alpha-Antagonists
  • Adrenergic beta-Antagonists
  • Antidepressive Agents
  • Carbon Isotopes
  • Catecholamines
  • Hallucinogens
  • Histamine H1 Antagonists
  • Monoamine Oxidase Inhibitors
  • Tranquilizing Agents
  • Serotonin
  • Histamine
  • Cyclic AMP
  • Isoproterenol
  • Norepinephrine
  • Epinephrine