Evidence for high and low affinity alpha 2-receptors. Comparison of [3H]norepinephrine and [3H]phentolamine binding to human platelet membranes

J Biol Chem. 1981 Apr 10;256(7):3298-303.
No abstract available

Publication types

  • Comparative Study
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Binding, Competitive
  • Blood Platelets / metabolism*
  • Cations, Monovalent
  • Cell Membrane / metabolism
  • Guanosine Triphosphate / pharmacology
  • Humans
  • Kinetics
  • Magnesium / pharmacology
  • Norepinephrine / blood*
  • Norepinephrine / pharmacology
  • Phentolamine / blood*
  • Receptors, Adrenergic / metabolism*
  • Receptors, Adrenergic, alpha / drug effects
  • Receptors, Adrenergic, alpha / metabolism*
  • Tritium

Substances

  • Cations, Monovalent
  • Receptors, Adrenergic
  • Receptors, Adrenergic, alpha
  • Tritium
  • Guanosine Triphosphate
  • Magnesium
  • Norepinephrine
  • Phentolamine