Assays for inhibitors of CAAX farnesyltransferase in vitro and in intact cells

Methods Enzymol. 1995:255:38-46. doi: 10.1016/s0076-6879(95)55007-0.
No abstract available

MeSH terms

  • Alkyl and Aryl Transferases*
  • Amino Acid Sequence
  • Animals
  • Baculoviridae / genetics
  • Brain / enzymology
  • Cells, Cultured
  • Enzyme Inhibitors / analysis
  • Escherichia coli / genetics
  • In Vitro Techniques
  • Molecular Sequence Data
  • Oligopeptides / analysis
  • Oligopeptides / chemistry
  • Oligopeptides / pharmacology
  • Rats
  • Recombinant Proteins / antagonists & inhibitors
  • Recombinant Proteins / genetics
  • Spodoptera
  • Transferases / antagonists & inhibitors*
  • Transferases / genetics

Substances

  • Enzyme Inhibitors
  • Oligopeptides
  • Recombinant Proteins
  • Transferases
  • Alkyl and Aryl Transferases
  • geranylgeranyltransferase type-I