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Novel xanthone-polyamine conjugates as catalytic inhibitors of human topoisomerase IIα.
Bioorg Med Chem Lett. 2017 Oct 15;27(20):4687-4693. doi: 10.1016/j.bmcl.2017.09.011. Epub 2017 Sep 8.
Bioorg Med Chem Lett. 2017.
PMID: 28919339
Free PMC article.
Pharmacophore Hybridization To Discover Novel Topoisomerase II Poisons with Promising Antiproliferative Activity.
Ortega JA, Riccardi L, Minniti E, Borgogno M, Arencibia JM, Greco ML, Minarini A, Sissi C, De Vivo M.
Ortega JA, et al. Among authors: minniti e.
J Med Chem. 2018 Feb 8;61(3):1375-1379. doi: 10.1021/acs.jmedchem.7b01388. Epub 2017 Nov 9.
J Med Chem. 2018.
PMID: 29077404
Free article.
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Benextramine and derivatives as novel human monoamine oxidases inhibitors: an integrated approach.
Di Paolo ML, Cozza G, Milelli A, Zonta F, Sarno S, Minniti E, Ursini F, Rosini M, Minarini A.
Di Paolo ML, et al. Among authors: minniti e.
FEBS J. 2019 Dec;286(24):4995-5015. doi: 10.1111/febs.14994. Epub 2019 Jul 29.
FEBS J. 2019.
PMID: 31291696
Free article.
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Novel, Potent, and Druglike Tetrahydroquinazoline Inhibitor That Is Highly Selective for Human Topoisomerase II α over β.
Ortega JA, Arencibia JM, Minniti E, Byl JAW, Franco-Ulloa S, Borgogno M, Genna V, Summa M, Bertozzi SM, Bertorelli R, Armirotti A, Minarini A, Sissi C, Osheroff N, De Vivo M.
Ortega JA, et al. Among authors: minniti e.
J Med Chem. 2020 Nov 12;63(21):12873-12886. doi: 10.1021/acs.jmedchem.0c00774. Epub 2020 Oct 20.
J Med Chem. 2020.
PMID: 33079544
Free PMC article.
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Polyamine-containing etoposide derivatives as poisons of human type II topoisomerases: Differential effects on topoisomerase IIα and IIβ.
Oviatt AA, Kuriappan JA, Minniti E, Vann KR, Onuorah P, Minarini A, De Vivo M, Osheroff N.
Oviatt AA, et al. Among authors: minniti e.
Bioorg Med Chem Lett. 2018 Sep 15;28(17):2961-2968. doi: 10.1016/j.bmcl.2018.07.010. Epub 2018 Jul 5.
Bioorg Med Chem Lett. 2018.
PMID: 30006062
Free PMC article.
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An optimized polyamine moiety boosts the potency of human type II topoisomerase poisons as quantified by comparative analysis centered on the clinical candidate F14512.
Palermo G, Minniti E, Greco ML, Riccardi L, Simoni E, Convertino M, Marchetti C, Rosini M, Sissi C, Minarini A, De Vivo M.
Palermo G, et al. Among authors: minniti e.
Chem Commun (Camb). 2015 Oct 1;51(76):14310-3. doi: 10.1039/c5cc05065k. Epub 2015 Aug 3.
Chem Commun (Camb). 2015.
PMID: 26234198
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