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hERG Optimization of Benzofuro-Pyridine and Pyrazino-Indole Derivatives as MCHR1 Antagonists.
ChemMedChem. 2022 Apr 5;17(7):e202100707. doi: 10.1002/cmdc.202100707. Epub 2022 Feb 3.
ChemMedChem. 2022.
PMID: 35041296
Design, synthesis and biological evaluation of novel cyclic malonamide derivatives as selective RIPK1 inhibitors.
Petró JL, Bényei G, Bana P, Linke N, Horti F, Szabó JE, Szalai KK, Hornyánszky G, Greiner I, Éles J.
Petró JL, et al. Among authors: szalai kk.
Bioorg Med Chem Lett. 2024 Mar 1;100:129643. doi: 10.1016/j.bmcl.2024.129643. Epub 2024 Feb 3.
Bioorg Med Chem Lett. 2024.
PMID: 38316369
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Aspartic acid scaffold in bradykinin B1 antagonists.
Huszár J, Timár Z, Bogár F, Penke B, Kiss R, Szalai KK, Schmidt E, Papp A, Keseru G.
Huszár J, et al. Among authors: szalai kk.
J Pept Sci. 2009 Jun;15(6):423-34. doi: 10.1002/psc.1134.
J Pept Sci. 2009.
PMID: 19378355
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Novel bradykinin-1 antagonists containing a (1,2,3,4-tetrahydro-isoquinolin-1-yl)acetic acid scaffold.
Huszár J, Timár Z, Szalai KK, Keseru G, Fülöp F, Penke B.
Huszár J, et al. Among authors: szalai kk.
Eur J Med Chem. 2008 Jul;43(7):1552-8. doi: 10.1016/j.ejmech.2007.10.030. Epub 2007 Nov 4.
Eur J Med Chem. 2008.
PMID: 18068274
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