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Non-peptide corticotropin-releasing hormone antagonists: syntheses and structure-activity relationships of 2-anilinopyrimidines and -triazines.
J Med Chem. 1999 Mar 11;42(5):805-18. doi: 10.1021/jm980222w.
J Med Chem. 1999.
PMID: 10072679
Corticotropin-releasing hormone receptor antagonists: framework design and synthesis guided by ligand conformational studies.
Hodge CN, Aldrich PE, Wasserman ZR, Fernandez CH, Nemeth GA, Arvanitis A, Cheeseman RS, Chorvat RJ, Ciganek E, Christos TE, Gilligan PJ, Krenitsky P, Scholfield E, Strucely P.
Hodge CN, et al. Among authors: krenitsky p.
J Med Chem. 1999 Mar 11;42(5):819-32. doi: 10.1021/jm980223o.
J Med Chem. 1999.
PMID: 10072680
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Synthesis, corticotropin-releasing factor receptor binding affinity, and pharmacokinetic properties of triazolo-, imidazo-, and pyrrolopyrimidines and -pyridines.
Chorvat RJ, Bakthavatchalam R, Beck JP, Gilligan PJ, Wilde RG, Cocuzza AJ, Hobbs FW, Cheeseman RS, Curry M, Rescinito JP, Krenitsky P, Chidester D, Yarem JA, Klaczkiewicz JD, Hodge CN, Aldrich PE, Wasserman ZR, Fernandez CH, Zaczek R, Fitzgerald LW, Huang SM, Shen HL, Wong YN, Chien BM, Arvanitis A, et al.
Chorvat RJ, et al. Among authors: krenitsky p.
J Med Chem. 1999 Mar 11;42(5):833-48. doi: 10.1021/jm980224g.
J Med Chem. 1999.
PMID: 10072681
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When structure-affinity relationships meet structure-kinetics relationships: 3-((Inden-1-yl)amino)-1-isopropyl-cyclopentane-1-carboxamides as CCR2 antagonists.
Vilums M, Zweemer AJ, Barmare F, van der Gracht AM, Bleeker DC, Yu Z, de Vries H, Gross R, Clemens J, Krenitsky P, Brussee J, Stamos D, Saunders J, Heitman LH, IJzerman AP.
Vilums M, et al.
Eur J Med Chem. 2015 Mar 26;93:121-34. doi: 10.1016/j.ejmech.2015.01.063. Epub 2015 Feb 2.
Eur J Med Chem. 2015.
PMID: 25666912
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Structure-kinetic relationships--an overlooked parameter in hit-to-lead optimization: a case of cyclopentylamines as chemokine receptor 2 antagonists.
Vilums M, Zweemer AJ, Yu Z, de Vries H, Hillger JM, Wapenaar H, Bollen IA, Barmare F, Gross R, Clemens J, Krenitsky P, Brussee J, Stamos D, Saunders J, Heitman LH, Ijzerman AP.
Vilums M, et al.
J Med Chem. 2013 Oct 10;56(19):7706-14. doi: 10.1021/jm4011737. Epub 2013 Sep 27.
J Med Chem. 2013.
PMID: 24028535
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Discovery of novel oxazepine and diazepine carboxamides as two new classes of heat shock protein 90 inhibitors.
Neubert T, Numa M, Ernst J, Clemens J, Krenitsky P, Liu M, Fleck B, Woody L, Zuccola H, Stamos D.
Neubert T, et al.
Bioorg Med Chem Lett. 2015 Mar 15;25(6):1338-42. doi: 10.1016/j.bmcl.2015.01.023. Epub 2015 Jan 20.
Bioorg Med Chem Lett. 2015.
PMID: 25677667
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Diastereoselective one-pot Knoevenagel condensation/Corey-Chaykovsky cyclopropanation.
Clemens JJ, Asgian JL, Busch BB, Coon T, Ernst J, Kaljevic L, Krenitsky PJ, Neubert TD, Schweiger EJ, Termin A, Stamos D.
Clemens JJ, et al. Among authors: krenitsky pj.
J Org Chem. 2013 Jan 18;78(2):780-5. doi: 10.1021/jo302443k. Epub 2012 Dec 31.
J Org Chem. 2013.
PMID: 23252964
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Orchestrated triple C-H activation reactions using two directing groups: rapid assembly of complex pyrazoles.
Yang W, Ye S, Fanning D, Coon T, Schmidt Y, Krenitsky P, Stamos D, Yu JQ.
Yang W, et al.
Angew Chem Int Ed Engl. 2015 Feb 16;54(8):2501-4. doi: 10.1002/anie.201410462. Epub 2015 Jan 16.
Angew Chem Int Ed Engl. 2015.
PMID: 25641121
Free PMC article.
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