Neumann U - Search Results

1

2-(diethylamino)thieno1,3ŏxazin-4-ones as stable inhibitors of human leukocyte elastase.

Gütschow M, Kuerschner L, Neumann U, Pietsch M, Löser R, Koglin N, Eger K. Gütschow M, et al. Among authors: neumann u. J Med Chem. 1999 Dec 30;42(26):5437-47. doi: 10.1021/jm991108w. J Med Chem. 1999. PMID: 10639285

2

Inhibition of cathepsin G by 4H-3,1-benzoxazin-4-ones.

Gütschow M, Neumann U. Gütschow M, et al. Among authors: neumann u. Bioorg Med Chem. 1997 Oct;5(10):1935-42. doi: 10.1016/s0968-0896(97)00128-4. Bioorg Med Chem. 1997. PMID: 9370038

3

Novel thieno[2,3-d][1,3]oxazin-4-ones as inhibitors of human leukocyte elastase.

Gütschow M, Neumann U. Gütschow M, et al. Among authors: neumann u. J Med Chem. 1998 May 7;41(10):1729-40. doi: 10.1021/jm9708341. J Med Chem. 1998. PMID: 9572899

4

Studies on 2-benzyloxy-4H-3,1-benzoxazin-4-ones as serine protease inhibitors.

Gütschow M, Neumann U, Sieler J, Eger K. Gütschow M, et al. Among authors: neumann u. Pharm Acta Helv. 1998 Jul;73(2):95-103. doi: 10.1016/s0031-6865(98)00003-x. Pharm Acta Helv. 1998. PMID: 9700938

5

Inhibition of human chymase by 2-amino-3,1-benzoxazin-4-ones.

Neumann U, Schechter NM, Gütschow M. Neumann U, et al. Bioorg Med Chem. 2001 Apr;9(4):947-54. doi: 10.1016/s0968-0896(00)00310-2. Bioorg Med Chem. 2001. PMID: 11354678

6

Inhibition of cathepsin G by 2-amino-3,1-benzoxazin-4-ones: kinetic investigations and docking studies.

Gütschow M, Kuerschner L, Pietsch M, Ambrozak A, Neumann U, Günther R, Hofmann HJ. Gütschow M, et al. Among authors: neumann u. Arch Biochem Biophys. 2002 Jun 15;402(2):180-91. doi: 10.1016/S0003-9861(02)00054-1. Arch Biochem Biophys. 2002. PMID: 12051662

7

N-(sulfonyloxy)phthalimides and analogues are potent inactivators of serine proteases.

Neumann U, Gütschow M. Neumann U, et al. J Biol Chem. 1994 Aug 26;269(34):21561-7. J Biol Chem. 1994. PMID: 8063794 Free article.

8

Synthesis of the Potent, Selective, and Efficacious β-Secretase (BACE1) Inhibitor NB-360.

Rueeger H, Lueoend R, Machauer R, Veenstra SJ, Holzer P, Hurth K, Voegtle M, Frederiksen M, Rondeau JM, Tintelnot-Blomley M, Jacobson LH, Staufenbiel M, Laue G, Neumann U. Rueeger H, et al. Among authors: neumann u. J Med Chem. 2021 Apr 22;64(8):4677-4696. doi: 10.1021/acs.jmedchem.0c02143. Epub 2021 Apr 12. J Med Chem. 2021. PMID: 33844524

9

Discovery of Umibecestat (CNP520): A Potent, Selective, and Efficacious β-Secretase (BACE1) Inhibitor for the Prevention of Alzheimer's Disease.

Machauer R, Lueoend R, Hurth K, Veenstra SJ, Rueeger H, Voegtle M, Tintelnot-Blomley M, Rondeau JM, Jacobson LH, Laue G, Beltz K, Neumann U. Machauer R, et al. Among authors: neumann u. J Med Chem. 2021 Oct 28;64(20):15262-15279. doi: 10.1021/acs.jmedchem.1c01300. Epub 2021 Oct 14. J Med Chem. 2021. PMID: 34648711

10

Inhibition of chymotrypsin and pancreatic elastase by 4H-3,1-benzoxazin-4-ones.

Neumann U, Stürzebecher J, Leistner S, Vieweg H. Neumann U, et al. J Enzyme Inhib. 1991;4(3):227-32. doi: 10.3109/14756369109035846. J Enzyme Inhib. 1991. PMID: 2037867

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