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Synthesis and pharmacological evaluation of new pyrazolidine-3, 5-diones as AT(1) angiotensin II receptor antagonists.
J Med Chem. 2000 Jul 13;43(14):2685-97. doi: 10.1021/jm9904147.
J Med Chem. 2000.
PMID: 10893306
Comparison of 3D structures and AT(1) binding properties of pyrazolidine-3,5-diones and tetrahydropyridazine-3,6-diones with parent antihypertensive drug irbesartan.
Le Bourdonnec B, Cauvin C, Meulon E, Yous S, Goossens JF, Durant F, Houssin R, Hénichart JP.
Le Bourdonnec B, et al. Among authors: meulon e.
J Med Chem. 2002 Oct 10;45(21):4794-8. doi: 10.1021/jm010457z.
J Med Chem. 2002.
PMID: 12361407
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