Zablocki JA - Search Results

1

Structure-affinity relationships of the affinity of 2-pyrazolyl adenosine analogues for the adenosine A2A receptor.

Palle VP, Elzein EO, Gothe SA, Li Z, Gao Z, Meyer S, Blackburn B, Zablocki JA. Palle VP, et al. Among authors: zablocki ja. Bioorg Med Chem Lett. 2002 Oct 21;12(20):2935-9. doi: 10.1016/s0960-894x(02)00609-1. Bioorg Med Chem Lett. 2002. PMID: 12270178

2

2-Pyrazolyl-N(6)-substituted adenosine derivatives as high affinity and selective adenosine A(3) receptor agonists.

Elzein E, Palle V, Wu Y, Maa T, Zeng D, Zablocki J. Elzein E, et al. J Med Chem. 2004 Sep 9;47(19):4766-73. doi: 10.1021/jm049682h. J Med Chem. 2004. PMID: 15341491

3

The discovery of a selective, high affinity A(2B) adenosine receptor antagonist for the potential treatment of asthma.

Zablocki J, Kalla R, Perry T, Palle V, Varkhedkar V, Xiao D, Piscopio A, Maa T, Gimbel A, Hao J, Chu N, Leung K, Zeng D. Zablocki J, et al. Bioorg Med Chem Lett. 2005 Feb 1;15(3):609-12. doi: 10.1016/j.bmcl.2004.11.044. Bioorg Med Chem Lett. 2005. PMID: 15664822

4

Novel 1,3-dipropyl-8-(1-heteroarylmethyl-1H-pyrazol-4-yl)-xanthine derivatives as high affinity and selective A2B adenosine receptor antagonists.

Elzein E, Kalla R, Li X, Perry T, Parkhill E, Palle V, Varkhedkar V, Gimbel A, Zeng D, Lustig D, Leung K, Zablocki J. Elzein E, et al. Bioorg Med Chem Lett. 2006 Jan 15;16(2):302-6. doi: 10.1016/j.bmcl.2005.10.002. Epub 2005 Nov 4. Bioorg Med Chem Lett. 2006. PMID: 16275090

5

Novel 1,3-disubstituted 8-(1-benzyl-1H-pyrazol-4-yl) xanthines: high affinity and selective A2B adenosine receptor antagonists.

Kalla RV, Elzein E, Perry T, Li X, Palle V, Varkhedkar V, Gimbel A, Maa T, Zeng D, Zablocki J. Kalla RV, et al. J Med Chem. 2006 Jun 15;49(12):3682-92. doi: 10.1021/jm051268+. J Med Chem. 2006. PMID: 16759111

6

N6-Cycloalkyl-2-substituted adenosine derivatives as selective, high affinity adenosine A1 receptor agonists.

Elzein E, Kalla R, Li X, Perry T, Marquart T, Micklatcher M, Li Y, Wu Y, Zeng D, Zablocki J. Elzein E, et al. Bioorg Med Chem Lett. 2007 Jan 1;17(1):161-6. doi: 10.1016/j.bmcl.2006.09.065. Epub 2006 Oct 11. Bioorg Med Chem Lett. 2007. PMID: 17045477

7

Selective, high affinity A(2B) adenosine receptor antagonists: N-1 monosubstituted 8-(pyrazol-4-yl)xanthines.

Kalla RV, Elzein E, Perry T, Li X, Gimbel A, Yang M, Zeng D, Zablocki J. Kalla RV, et al. Bioorg Med Chem Lett. 2008 Feb 15;18(4):1397-401. doi: 10.1016/j.bmcl.2008.01.008. Epub 2008 Jan 8. Bioorg Med Chem Lett. 2008. PMID: 18226896

8

Discovery of a novel A2B adenosine receptor antagonist as a clinical candidate for chronic inflammatory airway diseases.

Elzein E, Kalla RV, Li X, Perry T, Gimbel A, Zeng D, Lustig D, Leung K, Zablocki J. Elzein E, et al. J Med Chem. 2008 Apr 10;51(7):2267-78. doi: 10.1021/jm7014815. Epub 2008 Mar 6. J Med Chem. 2008. PMID: 18321039

9

Affinity and intrinsic efficacy (IE) of 5'-carbamoyl adenosine analogues for the A1 adenosine receptor--efforts towards the discovery of a chronic ventricular rate control agent for the treatment of atrial fibrillation (AF).

Palle VP, Varkhedkar V, Ibrahim P, Ahmed H, Li Z, Gao Z, Ozeck M, Wu Y, Zeng D, Wu L, Leung K, Chu N, Zablocki JA. Palle VP, et al. Among authors: zablocki ja. Bioorg Med Chem Lett. 2004 Jan 19;14(2):535-9. doi: 10.1016/j.bmcl.2003.09.094. Bioorg Med Chem Lett. 2004. PMID: 14698198

10

Structure-affinity relationships of 5'-aromatic ethers and 5'-aromatic sulfides as partial A1 adenosine agonists, potential supraventricular anti-arrhythmic agents.

Morrison CF, Elzein E, Jiang B, Ibrahim PN, Marquart T, Palle V, Shenk KD, Varkhedkar V, Maa T, Wu L, Wu Y, Zeng D, Fong I, Lustig D, Leung K, Zablocki JA. Morrison CF, et al. Among authors: zablocki ja. Bioorg Med Chem Lett. 2004 Jul 16;14(14):3793-7. doi: 10.1016/j.bmcl.2004.04.096. Bioorg Med Chem Lett. 2004. PMID: 15203164

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