Scarborough R - Search Results

1

Hydroxamate based inhibitors of adenylyl cyclase. Part 2: the effect of cyclic linkers on P-site binding.

Levy D, Bao M, Tomlinson J, Scarborough R. Levy D, et al. Among authors: scarborough r. Bioorg Med Chem Lett. 2002 Nov 4;12(21):3089-92. doi: 10.1016/s0960-894x(02)00654-6. Bioorg Med Chem Lett. 2002. PMID: 12372508

2

Hydroxamate based inhibitors of adenylyl cyclase. Part 1: the effect of acyclic linkers on P-site binding.

Levy D, Marlowe C, Kane-Maguire K, Bao M, Cherbavaz D, Tomlinson J, Sedlock D, Scarborough R. Levy D, et al. Among authors: scarborough r. Bioorg Med Chem Lett. 2002 Nov 4;12(21):3085-8. doi: 10.1016/s0960-894x(02)00653-4. Bioorg Med Chem Lett. 2002. PMID: 12372507

3

Metal coordination-based inhibitors of adenylyl cyclase: novel potent P-site antagonists.

Levy DE, Bao M, Cherbavaz DB, Tomlinson JE, Sedlock DM, Homcy CJ, Scarborough RM. Levy DE, et al. J Med Chem. 2003 May 22;46(11):2177-86. doi: 10.1021/jm0205604. J Med Chem. 2003. PMID: 12747789

4

Direct inhibition of type 5 adenylyl cyclase prevents myocardial apoptosis without functional deterioration.

Iwatsubo K, Minamisawa S, Tsunematsu T, Nakagome M, Toya Y, Tomlinson JE, Umemura S, Scarborough RM, Levy DE, Ishikawa Y. Iwatsubo K, et al. J Biol Chem. 2004 Sep 24;279(39):40938-45. doi: 10.1074/jbc.M314238200. Epub 2004 Jul 15. J Biol Chem. 2004. PMID: 15262973 Free article.

5

Design, synthesis, and SAR of substituted acrylamides as factor Xa inhibitors.

Song Y, Clizbe L, Bhakta C, Teng W, Li W, Wu Y, Jia ZJ, Zhang P, Wang L, Doughan B, Su T, Kanter J, Woolfrey J, Wong P, Huang B, Tran K, Sinha U, Park G, Reed A, Malinowski J, Hollenbach S, Scarborough RM, Zhu BY. Song Y, et al. Bioorg Med Chem Lett. 2002 Jun 3;12(11):1511-5. doi: 10.1016/s0960-894x(02)00199-3. Bioorg Med Chem Lett. 2002. PMID: 12031331

6

Design, synthesis and structure-activity relationships of benzoxazinone-based factor Xa inhibitors.

Huang W, Zhang P, Zuckett JF, Wang L, Woolfrey J, Song Y, Jia ZJ, Clizbe LA, Su T, Tran K, Huang B, Wong P, Sinha U, Park G, Reed A, Malinowski J, Hollenbach SJ, Scarborough RM, Zhu BY. Huang W, et al. Bioorg Med Chem Lett. 2003 Feb 10;13(3):561-6. doi: 10.1016/s0960-894x(02)00927-7. Bioorg Med Chem Lett. 2003. PMID: 12565972

7

Design, synthesis, and structure-activity relationships of substituted piperazinone-based transition state factor Xa inhibitors.

Su T, Yang H, Volkots D, Woolfrey J, Dam S, Wong P, Sinha U, Scarborough RM, Zhu BY. Su T, et al. Bioorg Med Chem Lett. 2003 Feb 24;13(4):729-32. doi: 10.1016/s0960-894x(02)01038-7. Bioorg Med Chem Lett. 2003. PMID: 12639568

8

Design, synthesis and biological activity of novel non-amidine factor Xa inhibitors. Part 1: P(1) structure-activity relationships of the substituted 1-(2-Naphthyl)-1H-pyrazole-5-carboxylamides.

Jia ZJ, Wu Y, Huang W, Goldman E, Zhang P, Woolfrey J, Wong P, Huang B, Sinha U, Park G, Reed A, Scarborough RM, Zhu BY. Jia ZJ, et al. Bioorg Med Chem Lett. 2002 Jun 17;12(12):1651-5. doi: 10.1016/s0960-894x(02)00239-1. Bioorg Med Chem Lett. 2002. PMID: 12039583

9

Parallel synthesis and structure-activity relationships of a series of highly potent, selective, and neutral factor Xa inhibitors.

Bauer SM, Goldman EA, Huang W, Su T, Wang L, Woolfrey J, Wu Y, Zuckett JF, Arfsten A, Huang B, Kothule J, Lin J, May B, Sinha U, Wong PW, Hutchaleelaha A, Scarborough RM, Zhu BY. Bauer SM, et al. Bioorg Med Chem Lett. 2004 Aug 2;14(15):4045-50. doi: 10.1016/j.bmcl.2004.05.033. Bioorg Med Chem Lett. 2004. PMID: 15225723

10

Design and synthesis of factor Xa inhibitors and their prodrugs.

Song Y, Clizbe L, Bhakta C, Teng W, Wong P, Huang B, Tran K, Sinha U, Park G, Reed A, Scarborough RM, Zhu BY. Song Y, et al. Bioorg Med Chem Lett. 2003 Jan 20;13(2):297-300. doi: 10.1016/s0960-894x(02)00921-6. Bioorg Med Chem Lett. 2003. PMID: 12482444

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