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New orally active PDE4 inhibitors with therapeutic potential.
Ochiai H, Ishida A, Ohtani T, Kusumi K, Kishikawa K, Obata T, Nakai H, Toda M. Ochiai H, et al. Among authors: kusumi k. Bioorg Med Chem Lett. 2004 Jan 5;14(1):29-32. doi: 10.1016/j.bmcl.2003.10.025. Bioorg Med Chem Lett. 2004. PMID: 14684291
Highly potent PDE4 inhibitors with therapeutic potential.
Ochiai H, Ohtani T, Ishida A, Kusumi K, Kato M, Kohno H, Kishikawa K, Obata T, Nakai H, Toda M. Ochiai H, et al. Among authors: kusumi k. Bioorg Med Chem Lett. 2004 Jan 5;14(1):207-10. doi: 10.1016/j.bmcl.2003.09.087. Bioorg Med Chem Lett. 2004. PMID: 14684329
New orally active PDE4 inhibitors with therapeutic potential.
Ochiai H, Ishida A, Ohtani T, Kusumi K, Kishikawa K, Yamamoto S, Takeda H, Obata T, Nakai H, Toda M. Ochiai H, et al. Among authors: kusumi k. Bioorg Med Chem. 2004 Aug 1;12(15):4089-100. doi: 10.1016/j.bmc.2004.05.032. Bioorg Med Chem. 2004. PMID: 15246087
Discovery of new orally active phosphodiesterase (PDE4) inhibitors.
Ochiai H, Ishida A, Ohtani T, Kusumi K, Kishikawa K, Yamamoto S, Takeda H, Obata T, Nakai H, Toda M. Ochiai H, et al. Among authors: kusumi k. Chem Pharm Bull (Tokyo). 2004 Sep;52(9):1098-104. doi: 10.1248/cpb.52.1098. Chem Pharm Bull (Tokyo). 2004. PMID: 15340197 Free article.
Highly potent PDE4 inhibitors with therapeutic potential.
Ochiai H, Ohtani T, Ishida A, Kusumi K, Kato M, Kohno H, Odagaki Y, Kishikawa K, Yamamoto S, Takeda H, Obata T, Nakai H, Toda M. Ochiai H, et al. Among authors: kusumi k. Bioorg Med Chem. 2004 Sep 1;12(17):4645-65. doi: 10.1016/j.bmc.2004.06.032. Bioorg Med Chem. 2004. PMID: 15358291
Discovery of S1P agonists with a dihydronaphthalene scaffold.
Kurata H, Kusumi K, Otsuki K, Suzuki R, Kurono M, Takada Y, Shioya H, Komiya T, Mizuno H, Ono T, Hagiya H, Minami M, Nakade S, Habashita H. Kurata H, et al. Among authors: kusumi k. Bioorg Med Chem Lett. 2011 Jul 1;21(13):3885-9. doi: 10.1016/j.bmcl.2011.05.029. Epub 2011 May 15. Bioorg Med Chem Lett. 2011. PMID: 21641216
Structure-activity relationship studies of S1P agonists with a dihydronaphthalene scaffold.
Kurata H, Kusumi K, Otsuki K, Suzuki R, Kurono M, Tokuda N, Takada Y, Shioya H, Mizuno H, Komiya T, Ono T, Hagiya H, Minami M, Nakade S, Habashita H. Kurata H, et al. Among authors: kusumi k. Bioorg Med Chem Lett. 2012 Jan 1;22(1):144-8. doi: 10.1016/j.bmcl.2011.11.048. Epub 2011 Nov 20. Bioorg Med Chem Lett. 2012. PMID: 22153936
143 results