Backfisch G - Search Results

1

Synthesis and SAR of highly potent and selective dopamine D3-receptor antagonists: variations on the 1H-pyrimidin-2-one theme.

Geneste H, Amberg W, Backfisch G, Beyerbach A, Braje WM, Delzer J, Haupt A, Hutchins CW, King LL, Sauer DR, Unger L, Wernet W. Geneste H, et al. Among authors: backfisch g. Bioorg Med Chem Lett. 2006 Apr 1;16(7):1934-7. doi: 10.1016/j.bmcl.2005.12.079. Epub 2006 Jan 24. Bioorg Med Chem Lett. 2006. PMID: 16439127

2

Synthesis and SAR of N-substituted dibenzazepinone derivatives as novel potent and selective alpha(V)beta(3) antagonists.

Kling A, Backfisch G, Delzer J, Geneste H, Graef C, Holzenkamp U, Hornberger W, Lange UE, Lauterbach A, Mack H, Seitz W, Subkowski T. Kling A, et al. Among authors: backfisch g. Bioorg Med Chem Lett. 2002 Feb 11;12(3):441-6. doi: 10.1016/s0960-894x(01)00773-9. Bioorg Med Chem Lett. 2002. PMID: 11814816

3

Synthesis of highly potent and selective hetaryl ureas as integrin alpha(V)beta3-receptor antagonists.

Lange UE, Backfisch G, Delzer J, Geneste H, Graef C, Hornberger W, Kling A, Lauterbach A, Subkowski T, Zechel C. Lange UE, et al. Among authors: backfisch g. Bioorg Med Chem Lett. 2002 May 20;12(10):1379-82. doi: 10.1016/s0960-894x(02)00161-0. Bioorg Med Chem Lett. 2002. PMID: 11992781

4

Highly potent and selective alphaVbeta3-receptor antagonists: solid-phase synthesis and SAR of 1-substituted 4-amino-1H-pyrimidin-2-ones.

Zechel C, Backfisch G, Delzer J, Geneste H, Graef C, Hornberger W, Kling A, Lange UE, Lauterbach A, Seitz W, Subkowski T. Zechel C, et al. Among authors: backfisch g. Bioorg Med Chem Lett. 2003 Jan 20;13(2):165-9. doi: 10.1016/s0960-894x(02)00931-9. Bioorg Med Chem Lett. 2003. PMID: 12482416

5

Design and synthesis of 1,5- and 2,5-substituted tetrahydrobenzazepinones as novel potent and selective integrin alphaVbeta3 antagonists.

Kling A, Backfisch G, Delzer J, Geneste H, Graef C, Hornberger W, Lange UE, Lauterbach A, Seitz W, Subkowski T. Kling A, et al. Among authors: backfisch g. Bioorg Med Chem. 2003 Apr 3;11(7):1319-41. doi: 10.1016/s0968-0896(02)00616-8. Bioorg Med Chem. 2003. PMID: 12628659

6

Synthesis and SAR of highly potent and selective dopamine D(3)-receptor antagonists: Quinolin(di)one and benzazepin(di)one derivatives. herve.geneste@abbott.com.

Geneste H, Backfisch G, Braje W, Delzer J, Haupt A, Hutchins CW, King LL, Lubisch W, Steiner G, Teschendorf HJ, Unger L, Wernet W. Geneste H, et al. Among authors: backfisch g. Bioorg Med Chem Lett. 2006 Feb;16(3):658-62. doi: 10.1016/j.bmcl.2005.10.035. Epub 2005 Nov 2. Bioorg Med Chem Lett. 2006. PMID: 16271293

7

Synthesis and SAR of highly potent and selective dopamine D(3)-receptor antagonists: 1H-pyrimidin-2-one derivatives.

Geneste H, Backfisch G, Braje W, Delzer J, Haupt A, Hutchins CW, King LL, Kling A, Teschendorf HJ, Unger L, Wernet W. Geneste H, et al. Among authors: backfisch g. Bioorg Med Chem Lett. 2006 Feb;16(3):490-4. doi: 10.1016/j.bmcl.2005.10.068. Epub 2005 Nov 11. Bioorg Med Chem Lett. 2006. PMID: 16290141

8

Design and synthesis of novel potent and selective integrin alphanubeta3 antagonists--novel synthetic routes to isoquinolinone, benzoxazinone, and quinazolinone acetates.

Seitz W, Geneste H, Backfisch G, Delzer J, Graef C, Hornberger W, Kling A, Subkowski T, Zimmermann N. Seitz W, et al. Among authors: backfisch g. Bioorg Med Chem Lett. 2008 Jan 15;18(2):527-31. doi: 10.1016/j.bmcl.2007.11.089. Epub 2007 Nov 28. Bioorg Med Chem Lett. 2008. PMID: 18068982

9

Potent and selective oxindole-based vasopressin 1b receptor antagonists with improved pharmacokinetic properties.

Oost T, Backfisch G, Bhowmik S, van Gaalen MM, Geneste H, Hornberger W, Lubisch W, Netz A, Unger L, Wernet W. Oost T, et al. Among authors: backfisch g. Bioorg Med Chem Lett. 2011 Jun 15;21(12):3828-31. doi: 10.1016/j.bmcl.2011.03.012. Epub 2011 Mar 6. Bioorg Med Chem Lett. 2011. PMID: 21605973

10

Mitigating the Metabolic Liability of Carbonyl Reduction: Novel Calpain Inhibitors with P1' Extension.

Kling A, Jantos K, Mack H, Hornberger W, Backfisch G, Lao Y, Nijsen M, Rendenbach-Mueller B, Moeller A. Kling A, et al. Among authors: backfisch g. ACS Med Chem Lett. 2018 Feb 4;9(3):221-226. doi: 10.1021/acsmedchemlett.7b00494. eCollection 2018 Mar 8. ACS Med Chem Lett. 2018. PMID: 29541364 Free PMC article.

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