Search Page
Save citations to file
Email citations
Send citations to clipboard
Add to Collections
Add to My Bibliography
Create a file for external citation management software
Your saved search
Your RSS Feed
Search Results
6 results
Filters applied: . Clear all
Results are displayed in a computed author sort order.
The Results By Year timeline is not available.
Page 1
Backbone cyclic peptidomimetic melanocortin-4 receptor agonist as a novel orally administrated drug lead for treating obesity.
J Med Chem. 2008 Feb 28;51(4):1026-34. doi: 10.1021/jm701093y. Epub 2008 Jan 26.
J Med Chem. 2008.
PMID: 18220330
Structure-activity relationship and metabolic stability studies of backbone cyclization and N-methylation of melanocortin peptides.
Linde Y, Ovadia O, Safrai E, Xiang Z, Portillo FP, Shalev DE, Haskell-Luevano C, Hoffman A, Gilon C.
Linde Y, et al. Among authors: portillo fp.
Biopolymers. 2008;90(5):671-82. doi: 10.1002/bip.21057.
Biopolymers. 2008.
PMID: 18655141
Free PMC article.
Item in Clipboard
Semi-rigid tripeptide agonists of melanocortin receptors.
Ruwe AR, Koikov L, Abdel-Malek Z, Haskell-Luevano C, Dirain ML, Portillo F, Xiang Z, Wortman M, Knittel JJ.
Ruwe AR, et al.
Bioorg Med Chem Lett. 2009 Sep 1;19(17):5176-81. doi: 10.1016/j.bmcl.2009.07.025. Epub 2009 Jul 9.
Bioorg Med Chem Lett. 2009.
PMID: 19635667
Free PMC article.
Item in Clipboard
Melanocortin tetrapeptide Ac-His-DPhe-Arg-Trp-NH2 modified at the para position of the benzyl side chain (DPhe): importance for mouse melanocortin-3 receptor agonist versus antagonist activity.
Proneth B, Pogozheva ID, Portillo FP, Mosberg HI, Haskell-Luevano C.
Proneth B, et al. Among authors: portillo fp.
J Med Chem. 2008 Sep 25;51(18):5585-93. doi: 10.1021/jm800291b.
J Med Chem. 2008.
PMID: 18800761
Free PMC article.
Item in Clipboard
A combination of ligand SAR and receptor site-directed mutagenesis reveals requirements for antagonist activity at the melanocortin-3 receptor.
Proneth B, Portillo FP, Haskell-Luevano C.
Proneth B, et al. Among authors: portillo fp.
Adv Exp Med Biol. 2009;611:319-20. doi: 10.1007/978-0-387-73657-0_142.
Adv Exp Med Biol. 2009.
PMID: 19400209
No abstract available.
Item in Clipboard
Discovery of Molecular Interactions of the Human Melanocortin-4 Receptor (hMC4R) Asp189 (D189) Amino Acid with the Endogenous G-Protein-Coupled Receptor (GPCR) Antagonist Agouti-Related Protein (AGRP) Provides Insights to AGRP's Inverse Agonist Pharmacology at the hMC4R.
Ericson MD, Haslach EM, Schnell SM, Freeman KT, Xiang ZM, Portillo FP, Speth R, Litherland SA, Haskell-Luevano C.
Ericson MD, et al. Among authors: portillo fp.
ACS Chem Neurosci. 2021 Feb 3;12(3):542-556. doi: 10.1021/acschemneuro.0c00755. Epub 2021 Jan 20.
ACS Chem Neurosci. 2021.
PMID: 33470098
Free PMC article.
Item in Clipboard
Cite
Cite