Kariv I - Search Results

1

Development of high-throughput TR-FRET and AlphaScreen assays for identification of potent inhibitors of PDK1.

Xu Z, Nagashima K, Sun D, Rush T, Northrup A, Andersen JN, Kariv I, Bobkova EV. Xu Z, et al. Among authors: kariv i. J Biomol Screen. 2009 Dec;14(10):1257-62. doi: 10.1177/1087057109349356. J Biomol Screen. 2009. PMID: 19822882

2

Efficient identification of novel leads by dynamic focused screening: PDK1 case stud.

Sun D, Jung J, Rush TS 3rd, Xu Z, Weber MJ, Bobkova E, Northrup A, Kariv I. Sun D, et al. Among authors: kariv i. Comb Chem High Throughput Screen. 2010 Jan;13(1):16-26. doi: 10.2174/138620710790218186. Comb Chem High Throughput Screen. 2010. PMID: 20214573

3

Discovery of PDK1 kinase inhibitors with a novel mechanism of action by ultrahigh throughput screening.

Bobkova EV, Weber MJ, Xu Z, Zhang YL, Jung J, Blume-Jensen P, Northrup A, Kunapuli P, Andersen JN, Kariv I. Bobkova EV, et al. Among authors: kariv i. J Biol Chem. 2010 Jun 11;285(24):18838-46. doi: 10.1074/jbc.M109.089946. Epub 2010 Apr 12. J Biol Chem. 2010. PMID: 20385558 Free PMC article.

4

Integration of Affinity Selection-Mass Spectrometry and Functional Cell-Based Assays to Rapidly Triage Druggable Target Space within the NF-κB Pathway.

Kutilek VD, Andrews CL, Richards MP, Xu Z, Sun T, Chen Y, Hashke A, Smotrov N, Fernandez R, Nickbarg EB, Chamberlin C, Sauvagnat B, Curran PJ, Boinay R, Saradjian P, Allen SJ, Byrne N, Elsen NL, Ford RE, Hall DL, Kornienko M, Rickert KW, Sharma S, Shipman JM, Lumb KJ, Coleman K, Dandliker PJ, Kariv I, Beutel B. Kutilek VD, et al. Among authors: kariv i. J Biomol Screen. 2016 Jul;21(6):608-19. doi: 10.1177/1087057116637353. Epub 2016 Mar 11. J Biomol Screen. 2016. PMID: 26969322

5

Development of High-Throughput Assays for Evaluation of Hematopoietic Progenitor Kinase 1 Inhibitors.

Lacey BM, Xu Z, Chai X, Laskey J, Fradera X, Mittal P, Mishra S, Piesvaux J, Saradjian P, Shaffer L, Vassileva G, Gerdt C, Wang Y, Ferguson H, Smith DM, Ballard J, Wells S, Jain R, Mueller U, Addona G, Kariv I, Methot JL, Bittinger M, Ranganath S, Mcleod R, Pasternak A, Miller JR, Xu H. Lacey BM, et al. Among authors: kariv i. SLAS Discov. 2021 Jan;26(1):88-99. doi: 10.1177/2472555220952071. Epub 2020 Aug 26. SLAS Discov. 2021. PMID: 32844715 Free article.

6

Development of a cell-based assay for measurement of c-Met phosphorylation using AlphaScreen technology and high-content imaging analysis.

Smotrov N, Mathur A, Kariv I, Moxham CM, Bays N. Smotrov N, et al. Among authors: kariv i. J Biomol Screen. 2009 Apr;14(4):404-11. doi: 10.1177/1087057109331803. J Biomol Screen. 2009. PMID: 19403923

7

Identification of inhibitors of bacterial transcription/translation machinery utilizing a miniaturized 1536-well format screen.

Kariv I, Cao H, Marvil PD, Bobkova EV, Bukhtiyarov YE, Yan YP, Patel U, Coudurier L, Chung TD, Oldenburg KR. Kariv I, et al. J Biomol Screen. 2001 Aug;6(4):233-43. doi: 10.1177/108705710100600405. J Biomol Screen. 2001. PMID: 11689123

8

A simplified scintillation proximity assay for fatty acid synthase activity: development and comparison with other FAS activity assays.

Bays NW, Hill AD, Kariv I. Bays NW, et al. Among authors: kariv i. J Biomol Screen. 2009 Jul;14(6):636-42. doi: 10.1177/1087057109335746. Epub 2009 Jun 16. J Biomol Screen. 2009. PMID: 19531664

9

Establishing and Validating Cellular Functional Target Engagement Assay for Selective IRAK4 Inhibitor Discovery.

Chen Y, Sun D, Yang R, Lim J, Sondey C, Presland J, Rakhilina L, Addona G, Kariv I, Chen H. Chen Y, et al. Among authors: kariv i. SLAS Discov. 2021 Sep;26(8):1040-1054. doi: 10.1177/24725552211021074. Epub 2021 Jun 16. SLAS Discov. 2021. PMID: 34130529 Free article.

10

High-throughput analysis of HGF-stimulated cell scattering.

Chan GK, Lutterbach BA, Pan BS, Kariv I, Szewczak AA. Chan GK, et al. Among authors: kariv i. J Biomol Screen. 2008 Oct;13(9):847-54. doi: 10.1177/1087057108324497. Epub 2008 Sep 23. J Biomol Screen. 2008. PMID: 18812567

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