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Page 1
Structure-activity relationships of 6-methyl-benzo[b]thiophene-2-carboxylic acid (1-[(S)-1-benzyl-4-[4-(tetrahydropyran-4-ylmethyl)piperazin-1-yl]butylcarbamoyl]cyclopentyl)amide, potent antagonist of the neurokinin-2 receptor.
Fattori D, Porcelloni M, D'Andrea P, Catalioto RM, Ettorre A, Giuliani S, Marastoni E, Mauro S, Meini S, Rossi C, Altamura M, Maggi CA. Fattori D, et al. Among authors: mauro s. J Med Chem. 2010 May 27;53(10):4148-65. doi: 10.1021/jm100176s. J Med Chem. 2010. PMID: 20408549
Alkyl piperidine and piperazine hydroxamic acids as HDAC inhibitors.
Rossi C, Porcelloni M, D'Andrea P, Fincham CI, Ettorre A, Mauro S, Squarcia A, Bigioni M, Parlani M, Nardelli F, Binaschi M, Maggi CA, Fattori D. Rossi C, et al. Among authors: mauro s. Bioorg Med Chem Lett. 2011 Apr 15;21(8):2305-8. doi: 10.1016/j.bmcl.2011.02.085. Epub 2011 Feb 26. Bioorg Med Chem Lett. 2011. PMID: 21420859
4-N-Hydroxy-4-[1-(sulfonyl)piperidin-4-yl]-butyramides as HDAC inhibitors.
Rossi C, Fincham CI, D'Andrea P, Porcelloni M, Ettorre A, Mauro S, Bigioni M, Binaschi M, Maggi CA, Nardelli F, Parlani M, Fattori D. Rossi C, et al. Among authors: mauro s. Bioorg Med Chem Lett. 2011 Nov 15;21(22):6767-9. doi: 10.1016/j.bmcl.2011.09.042. Epub 2011 Sep 18. Bioorg Med Chem Lett. 2011. PMID: 21978679
Design and synthesis of novel sulfonamide-containing bradykinin hB(2) receptor antagonists. Synthesis and structure-relationships of α,α-tetrahydropyranylglycine.
Fincham CI, Bressan A, D'Andrea P, Ettorre A, Giuliani S, Mauro S, Meini S, Paris M, Quartara L, Rossi C, Squarcia A, Valenti C, Daniela F, Maggi CA. Fincham CI, et al. Among authors: mauro s. Bioorg Med Chem. 2012 Mar 15;20(6):2091-100. doi: 10.1016/j.bmc.2012.01.036. Epub 2012 Jan 30. Bioorg Med Chem. 2012. PMID: 22342268
Benzofused hydroxamic acids: useful fragments for the preparation of histone deacetylase inhibitors. Part 2: 7-fluorobenzothiophenes and benzofurans.
Marastoni E, Bartoli S, Berettoni M, Cipollone A, Ettorre A, Fincham CI, Mauro S, Paris M, Porcelloni M, Bigioni M, Binaschi M, Nardelli F, Parlani M, Maggi CA, Paoli P, Rossi P, Fattori D. Marastoni E, et al. Among authors: mauro s. Bioorg Med Chem Lett. 2015 Apr 1;25(7):1603-6. doi: 10.1016/j.bmcl.2015.02.007. Epub 2015 Feb 24. Bioorg Med Chem Lett. 2015. PMID: 25746815
Benzofused hydroxamic acids: useful fragments for the preparation of histone deacetylase inhibitors. Part 1: hit identification.
Marastoni E, Bartoli S, Berettoni M, Cipollone A, Ettorre A, Fincham CI, Mauro S, Paris M, Porcelloni M, Bigioni M, Binaschi M, Nardelli F, Parlani M, Maggi CA, Fattori D. Marastoni E, et al. Among authors: mauro s. Bioorg Med Chem Lett. 2013 Jul 15;23(14):4091-5. doi: 10.1016/j.bmcl.2013.05.053. Epub 2013 May 25. Bioorg Med Chem Lett. 2013. PMID: 23768910
326 results