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Selective angiotensin II AT(2) receptor agonists with reduced CYP 450 inhibition.
Bioorg Med Chem. 2010 Jun 15;18(12):4570-90. doi: 10.1016/j.bmc.2010.03.064. Epub 2010 Apr 9.
Bioorg Med Chem. 2010.
PMID: 20493713
Selective angiotensin II AT2 receptor agonists: arylbenzylimidazole structure-activity relationships.
Wu X, Wan Y, Mahalingam AK, Murugaiah AM, Plouffe B, Botros M, Karlén A, Hallberg M, Gallo-Payet N, Alterman M.
Wu X, et al. Among authors: murugaiah am.
J Med Chem. 2006 Nov 30;49(24):7160-8. doi: 10.1021/jm0606185.
J Med Chem. 2006.
PMID: 17125268
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Selective angiotensin II AT(2) receptor agonists devoid of the imidazole ring system.
Murugaiah AM, Wallinder C, Mahalingam AK, Wu X, Wan Y, Plouffe B, Botros M, Karlén A, Hallberg M, Gallo-Payet N, Alterman M.
Murugaiah AM, et al.
Bioorg Med Chem. 2007 Nov 15;15(22):7166-83. doi: 10.1016/j.bmc.2007.07.026. Epub 2007 Aug 22.
Bioorg Med Chem. 2007.
PMID: 17825570
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From the first selective non-peptide AT(2) receptor agonist to structurally related antagonists.
Murugaiah AM, Wu X, Wallinder C, Mahalingam AK, Wan Y, Sköld C, Botros M, Guimond MO, Joshi A, Nyberg F, Gallo-Payet N, Hallberg A, Alterman M.
Murugaiah AM, et al.
J Med Chem. 2012 Mar 8;55(5):2265-78. doi: 10.1021/jm2015099. Epub 2012 Feb 22.
J Med Chem. 2012.
PMID: 22248302
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