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Discovery of 2-aminoimidazopyridine adenosine A(2A) receptor antagonists.
Bioorg Med Chem Lett. 2010 Nov 15;20(22):6845-9. doi: 10.1016/j.bmcl.2010.08.064. Epub 2010 Aug 19.
Bioorg Med Chem Lett. 2010.
PMID: 20869242
Novel pyrrolidine heterocycles as CCR1 antagonists.
Merritt JR, James R, Paradkar VM, Zhang C, Liu R, Liu J, Jacob B, Chiriac C, Ohlmeyer MJ, Quadros E, Wines P, Postelnek J, Hicks CM, Chen W, Kimble EF, O'Brien L, White N, Desai H, Appell KC, Webb ML.
Merritt JR, et al.
Bioorg Med Chem Lett. 2010 Sep 15;20(18):5477-9. doi: 10.1016/j.bmcl.2010.07.082. Epub 2010 Jul 24.
Bioorg Med Chem Lett. 2010.
PMID: 20708929
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Characterization of RWJ-351647, a novel nonpeptide vasopressin V2 receptor antagonist.
Gunnet JW, Matthews JM, Maryanoff BE, de Garavilla L, Andrade-Gordon P, Damiano B, Hageman W, Look R, Stahle P, Streeter AJ, Wines PG, Demarest KT.
Gunnet JW, et al. Among authors: wines pg.
Clin Exp Pharmacol Physiol. 2006 Apr;33(4):320-6. doi: 10.1111/j.1440-1681.2006.04369.x.
Clin Exp Pharmacol Physiol. 2006.
PMID: 16620295
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Pharmacological characterization of RWJ-676070, a dual vasopressin V(1A)/V(2) receptor antagonist.
Gunnet JW, Wines P, Xiang M, Rybczynski P, Andrade-Gordon P, de Garavilla L, Parry TJ, Cheung WM, Minor L, Demarest KT, Maryanoff BE, Damiano BP.
Gunnet JW, et al.
Eur J Pharmacol. 2008 Aug 20;590(1-3):333-42. doi: 10.1016/j.ejphar.2008.06.010. Epub 2008 Jun 7.
Eur J Pharmacol. 2008.
PMID: 18599033
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Enhancement of arachidonic acid signaling pathway by nicotinic acid receptor HM74A.
Tang Y, Zhou L, Gunnet JW, Wines PG, Cryan EV, Demarest KT.
Tang Y, et al. Among authors: wines pg.
Biochem Biophys Res Commun. 2006 Jun 23;345(1):29-37. doi: 10.1016/j.bbrc.2006.04.051. Epub 2006 Apr 25.
Biochem Biophys Res Commun. 2006.
PMID: 16674924
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