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Potent and selective HIV-1 ribonuclease H inhibitors based on a 1-hydroxy-1,8-naphthyridin-2(1H)-one scaffold.
Bioorg Med Chem Lett. 2010 Nov 15;20(22):6754-7. doi: 10.1016/j.bmcl.2010.08.135. Epub 2010 Sep 24.
Bioorg Med Chem Lett. 2010.
PMID: 20869872
Substituted tetrahydroquinolines as potent allosteric inhibitors of reverse transcriptase and its key mutants.
Su DS, Lim JJ, Tinney E, Wan BL, Young MB, Anderson KD, Rudd D, Munshi V, Bahnck C, Felock PJ, Lu M, Lai MT, Touch S, Moyer G, Distefano DJ, Flynn JA, Liang Y, Sanchez R, Prasad S, Yan Y, Perlow-Poehnelt R, Torrent M, Miller M, Vacca JP, Williams TM, Anthony NJ.
Su DS, et al.
Bioorg Med Chem Lett. 2009 Sep 1;19(17):5119-23. doi: 10.1016/j.bmcl.2009.07.031. Epub 2009 Jul 10.
Bioorg Med Chem Lett. 2009.
PMID: 19631528
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Biaryl ethers as potent allosteric inhibitors of reverse transcriptase and its key mutant viruses: aryl substituted pyrazole as a surrogate for the pyrazolopyridine motif.
Su DS, Lim JJ, Tinney E, Tucker TJ, Saggar S, Sisko JT, Wan BL, Young MB, Anderson KD, Rudd D, Munshi V, Bahnck C, Felock PJ, Lu M, Lai MT, Touch S, Moyer G, Distefano DJ, Flynn JA, Liang Y, Sanchez R, Perlow-Poehnelt R, Miller M, Vacca JP, Williams TM, Anthony NJ.
Su DS, et al.
Bioorg Med Chem Lett. 2010 Aug 1;20(15):4328-32. doi: 10.1016/j.bmcl.2010.06.083. Epub 2010 Jun 17.
Bioorg Med Chem Lett. 2010.
PMID: 20609585
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Biaryl ethers as novel non-nucleoside reverse transcriptase inhibitors with improved potency against key mutant viruses.
Su DS, Lim JJ, Tinney E, Wan BL, Young MB, Anderson KD, Rudd D, Munshi V, Bahnck C, Felock PJ, Lu M, Lai MT, Touch S, Moyer G, DiStefano DJ, Flynn JA, Liang Y, Sanchez R, Perlow-Poehnelt R, Miller M, Vacca JP, Williams TM, Anthony NJ.
Su DS, et al.
J Med Chem. 2009 Nov 26;52(22):7163-9. doi: 10.1021/jm901230r.
J Med Chem. 2009.
PMID: 19883100
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Development of a sensitive amplified luminescent proximity homogeneous assay to monitor the interactions between pTEFb and Tat.
Burlein C, Bahnck C, Bhatt T, Murphy D, Lemaire P, Carroll S, Miller MD, Lai MT.
Burlein C, et al.
Anal Biochem. 2014 Nov 15;465:164-71. doi: 10.1016/j.ab.2014.08.007. Epub 2014 Aug 14.
Anal Biochem. 2014.
PMID: 25132562
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Chondroitin sulfate promotes activation of cathepsin K.
Lemaire PA, Huang L, Zhuo Y, Lu J, Bahnck C, Stachel SJ, Carroll SS, Duong LT.
Lemaire PA, et al.
J Biol Chem. 2014 Aug 1;289(31):21562-72. doi: 10.1074/jbc.M114.559898. Epub 2014 Jun 23.
J Biol Chem. 2014.
PMID: 24958728
Free PMC article.
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Rapid assay to identify the two genetic forms of Culex (Culex) pipiens L. (Diptera: Culicidae) and hybrid populations.
Bahnck CM, Fonseca DM.
Bahnck CM, et al.
Am J Trop Med Hyg. 2006 Aug;75(2):251-5.
Am J Trop Med Hyg. 2006.
PMID: 16896127
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Dietary Ethanol Mediates Selection on Aldehyde Dehydrogenase Activity in Drosophila melanogaster.
Fry JD, Bahnck CM, Mikucki M, Phadnis N, Slattery WC.
Fry JD, et al. Among authors: bahnck cm.
Integr Comp Biol. 2004 Aug;44(4):275-83. doi: 10.1093/icb/44.4.275.
Integr Comp Biol. 2004.
PMID: 21676710
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