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Integration of lead optimization with crystallography for a membrane-bound ion channel target: discovery of a new class of AMPA receptor positive allosteric modulators.
J Med Chem. 2011 Jan 13;54(1):78-94. doi: 10.1021/jm100679e. Epub 2010 Dec 3.
J Med Chem. 2011.
PMID: 21128618
Discovery of N-[(2S)-5-(6-fluoro-3-pyridinyl)-2,3-dihydro-1H-inden-2-yl]-2-propanesulfonamide, a novel clinical AMPA receptor positive modulator.
Ward SE, Harries M, Aldegheri L, Andreotti D, Ballantine S, Bax BD, Harris AJ, Harker AJ, Lund J, Melarange R, Mingardi A, Mookherjee C, Mosley J, Neve M, Oliosi B, Profeta R, Smith KJ, Smith PW, Spada S, Thewlis KM, Yusaf SP.
Ward SE, et al. Among authors: mookherjee c.
J Med Chem. 2010 Aug 12;53(15):5801-12. doi: 10.1021/jm1005429.
J Med Chem. 2010.
PMID: 20614889
Clinical Trial.
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N-substituted pyrrolidines and tetrahydrofurans as novel AMPAR positive modulators.
Thewlis KM, Aldegheri L, Harries MH, Mookherjee C, Oliosi B, Ward SE.
Thewlis KM, et al. Among authors: mookherjee c.
Bioorg Med Chem Lett. 2010 Dec 1;20(23):7116-9. doi: 10.1016/j.bmcl.2010.09.062. Epub 2010 Sep 17.
Bioorg Med Chem Lett. 2010.
PMID: 20971003
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Identification of a sulfonamide series of CCR2 antagonists.
Peace S, Philp J, Brooks C, Piercy V, Moores K, Smethurst C, Watson S, Gaines S, Zippoli M, Mookherjee C, Ife R.
Peace S, et al. Among authors: mookherjee c.
Bioorg Med Chem Lett. 2010 Jul 1;20(13):3961-4. doi: 10.1016/j.bmcl.2010.04.142. Epub 2010 May 7.
Bioorg Med Chem Lett. 2010.
PMID: 20627722
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In vivo activity of an azole series of CCR2 antagonists.
Smethurst CA, Bevan N, Brooks C, Emmons A, Gough PJ, Mookherjee C, Moores K, Peace S, Philp J, Piercy V, Watson SP, Zippoli M.
Smethurst CA, et al. Among authors: mookherjee c.
Bioorg Med Chem Lett. 2012 Dec 1;22(23):7252-5. doi: 10.1016/j.bmcl.2012.09.020. Epub 2012 Sep 23.
Bioorg Med Chem Lett. 2012.
PMID: 23079519
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The discovery of a series of N-substituted 3-(4-piperidinyl)-1,3-benzoxazolinones and oxindoles as highly brain penetrant, selective muscarinic M1 agonists.
Johnson DJ, Forbes IT, Watson SP, Garzya V, Stevenson GI, Walker GR, Mudhar HS, Flynn ST, Wyman PA, Smith PW, Murkitt GS, Lucas AJ, Mookherjee CR, Watson JM, Gartlon JE, Bradford AM, Brown F.
Johnson DJ, et al. Among authors: mookherjee cr.
Bioorg Med Chem Lett. 2010 Sep 15;20(18):5434-8. doi: 10.1016/j.bmcl.2010.07.097. Epub 2010 Jul 30.
Bioorg Med Chem Lett. 2010.
PMID: 20709550
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The PPARdelta agonist GW0742X reduces atherosclerosis in LDLR(-/-) mice.
Graham TL, Mookherjee C, Suckling KE, Palmer CN, Patel L.
Graham TL, et al. Among authors: mookherjee c.
Atherosclerosis. 2005 Jul;181(1):29-37. doi: 10.1016/j.atherosclerosis.2004.12.028.
Atherosclerosis. 2005.
PMID: 15939051
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The characterisation of the major metabolite of salmeterol in the dog.
Bowers GD, Bayliss MK, Donnelly MC, Fellows I, Ismail IM, Mookherjee CR.
Bowers GD, et al. Among authors: mookherjee cr.
J Pharm Biomed Anal. 1998 Nov;18(3):461-70. doi: 10.1016/s0731-7085(98)00114-9.
J Pharm Biomed Anal. 1998.
PMID: 10096840
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