Matasi JJ - Search Results

1

Synthesis and SAR development of novel P2X7 receptor antagonists for the treatment of pain: part 1.

Matasi JJ, Brumfield S, Tulshian D, Czarnecki M, Greenlee W, Garlisi CG, Qiu H, Devito K, Chen SC, Sun Y, Bertorelli R, Geiss W, Le VD, Martin GS, Vellekoop SA, Haber J, Allard ML. Matasi JJ, et al. Bioorg Med Chem Lett. 2011 Jun 15;21(12):3805-8. doi: 10.1016/j.bmcl.2011.04.034. Epub 2011 Apr 24. Bioorg Med Chem Lett. 2011. PMID: 21570840

2

Structure-activity relationships of 2,4-diphenyl-1H-imidazole analogs as CB2 receptor agonists for the treatment of chronic pain.

Yang SW, Smotryski J, Matasi J, Ho G, Tulshian D, Greenlee WJ, Brusa R, Beltramo M, Cox K. Yang SW, et al. Bioorg Med Chem Lett. 2011 Jan 1;21(1):182-5. doi: 10.1016/j.bmcl.2010.11.044. Epub 2010 Nov 11. Bioorg Med Chem Lett. 2011. PMID: 21115245

3

Discovery of pyrrolo-benzo-1,4-diazines as potent Na(v)1.7 sodium channel blockers.

Ho GD, Tulshian D, Bercovici A, Tan Z, Hanisak J, Brumfield S, Matasi J, Heap CR, Earley WG, Courneya B, Herr RJ, Zhou X, Bridal T, Rindgen D, Sorota S, Yang SW. Ho GD, et al. Bioorg Med Chem Lett. 2014 Sep 1;24(17):4110-3. doi: 10.1016/j.bmcl.2014.07.060. Epub 2014 Jul 29. Bioorg Med Chem Lett. 2014. PMID: 25113934

4

Bioavailable pyrrolo-benzo-1,4-diazines as Na(v)1.7 sodium channel blockers for the treatment of pain.

Yang SW, Ho GD, Tulshian D, Bercovici A, Tan Z, Hanisak J, Brumfield S, Matasi J, Sun X, Sakwa SA, Herr RJ, Zhou X, Bridal T, Urban M, Vivian J, Rindgen D, Sorota S. Yang SW, et al. Bioorg Med Chem Lett. 2014 Nov 1;24(21):4958-62. doi: 10.1016/j.bmcl.2014.09.038. Epub 2014 Sep 19. Bioorg Med Chem Lett. 2014. PMID: 25288187

5

Initial optimization and series evolution of diaminopyrimidine inhibitors of interleukin-1 receptor associated kinase 4.

Seganish WM, McElroy WT, Herr RJ, Brumfield S, Greenlee WJ, Harding J, Komanduri V, Matasi J, Prakash KC, Tulshian D, Yang J, Yet L, Devito K, Fossetta J, Garlisi CG, Lundell D, Niu X, Sondey C. Seganish WM, et al. Bioorg Med Chem Lett. 2015 Aug 15;25(16):3203-7. doi: 10.1016/j.bmcl.2015.05.097. Epub 2015 Jun 6. Bioorg Med Chem Lett. 2015. PMID: 26115573

6

The discovery and synthesis of novel adenosine receptor (A(2A)) antagonists.

Matasi JJ, Caldwell JP, Hao J, Neustadt B, Arik L, Foster CJ, Lachowicz J, Tulshian DB. Matasi JJ, et al. Bioorg Med Chem Lett. 2005 Mar 1;15(5):1333-6. doi: 10.1016/j.bmcl.2005.01.019. Bioorg Med Chem Lett. 2005. PMID: 15713381

7

2-(2-Furanyl)-7-phenyl[1,2,4]triazolo[1,5-c]pyrimidin-5-amine analogs: highly potent, orally active, adenosine A2A antagonists. Part 1.

Matasi JJ, Caldwell JP, Zhang H, Fawzi A, Cohen-Williams ME, Varty GB, Tulshian DB. Matasi JJ, et al. Bioorg Med Chem Lett. 2005 Aug 15;15(16):3670-4. doi: 10.1016/j.bmcl.2005.05.086. Bioorg Med Chem Lett. 2005. PMID: 15978806

8

2-(2-Furanyl)-7-phenyl[1,2,4]triazolo[1,5-c]pyrimidin-5-amine analogs as adenosine A2A antagonists: the successful reduction of hERG activity. Part 2.

Matasi JJ, Caldwell JP, Zhang H, Fawzi A, Higgins GA, Cohen-Williams ME, Varty GB, Tulshian DB. Matasi JJ, et al. Bioorg Med Chem Lett. 2005 Aug 15;15(16):3675-8. doi: 10.1016/j.bmcl.2005.05.043. Bioorg Med Chem Lett. 2005. PMID: 15982882

9

3H-[1,2,4]-Triazolo[5,1-i]purin-5-amine derivatives as adenosine A2A antagonists.

Silverman LS, Caldwell JP, Greenlee WJ, Kiselgof E, Matasi JJ, Tulshian DB, Arik L, Foster C, Bertorelli R, Monopoli A, Ongini E. Silverman LS, et al. Among authors: matasi jj. Bioorg Med Chem Lett. 2007 Mar 15;17(6):1659-62. doi: 10.1016/j.bmcl.2006.12.104. Epub 2007 Jan 8. Bioorg Med Chem Lett. 2007. PMID: 17234414

10

Synthesis and structure-activity relationships of N-substituted spiropiperidines as nociceptin receptor ligands.

Caldwell JP, Matasi JJ, Zhang H, Fawzi A, Tulshian DB. Caldwell JP, et al. Among authors: matasi jj. Bioorg Med Chem Lett. 2007 Apr 15;17(8):2281-4. doi: 10.1016/j.bmcl.2007.01.069. Epub 2007 Jan 27. Bioorg Med Chem Lett. 2007. PMID: 17289383

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

21 results

Search Page