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Novel potent dual inhibitors of CK2 and Pim kinases with antiproliferative activity against cancer cells.
Bioorg Med Chem Lett. 2012 May 1;22(9):3327-31. doi: 10.1016/j.bmcl.2012.02.099. Epub 2012 Mar 6.
Bioorg Med Chem Lett. 2012.
PMID: 22460033
7-(4H-1,2,4-Triazol-3-yl)benzo[c][2,6]naphthyridines: a novel class of Pim kinase inhibitors with potent cell antiproliferative activity.
Pierre F, Stefan E, Nédellec AS, Chevrel MC, Regan CF, Siddiqui-Jain A, Macalino D, Streiner N, Drygin D, Haddach M, O'Brien SE, Anderes K, Ryckman DM.
Pierre F, et al. Among authors: regan cf.
Bioorg Med Chem Lett. 2011 Nov 15;21(22):6687-92. doi: 10.1016/j.bmcl.2011.09.059. Epub 2011 Sep 22.
Bioorg Med Chem Lett. 2011.
PMID: 21982499
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Synthesis and SAR of inhibitors of protein kinase CK2: novel tricyclic quinoline analogs.
Haddach M, Pierre F, Regan CF, Borsan C, Michaux J, Stefan E, Kerdoncuff P, Schwaebe MK, Chua PC, Siddiqui-Jain A, Macalino D, Drygin D, O'Brien SE, Rice WG, Ryckman DM.
Haddach M, et al. Among authors: regan cf.
Bioorg Med Chem Lett. 2012 Jan 1;22(1):45-8. doi: 10.1016/j.bmcl.2011.11.087. Epub 2011 Nov 30.
Bioorg Med Chem Lett. 2012.
PMID: 22169261
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Potent, orally active corticotropin-releasing factor receptor-1 antagonists containing a tricyclic pyrrolopyridine or pyrazolopyridine core.
Dyck B, Grigoriadis DE, Gross RS, Guo Z, Haddach M, Marinkovic D, McCarthy JR, Moorjani M, Regan CF, Saunders J, Schwaebe MK, Szabo T, Williams JP, Zhang X, Bozigian H, Chen TK.
Dyck B, et al. Among authors: regan cf.
J Med Chem. 2005 Jun 16;48(12):4100-10. doi: 10.1021/jm050070m.
J Med Chem. 2005.
PMID: 15943483
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Structure-activity relationships of 1,3,5-triazine-2,4,6-triones as human gonadotropin-releasing hormone receptor antagonists.
Guo Z, Wu D, Zhu YF, Tucci FC, Regan CF, Rowbottom MW, Struthers RS, Xie Q, Reijmers S, Sullivan SK, Sai Y, Chen C.
Guo Z, et al. Among authors: regan cf.
Bioorg Med Chem Lett. 2005 Aug 15;15(16):3685-90. doi: 10.1016/j.bmcl.2005.05.038.
Bioorg Med Chem Lett. 2005.
PMID: 15951171
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Se-phenyl prop-2-eneselenoate: an ethylene equivalent for Diels-Alder reactions.
Jung ME, Perez F, Regan CF, Yi SW, Perron Q.
Jung ME, et al. Among authors: regan cf.
Angew Chem Int Ed Engl. 2013 Feb 11;52(7):2060-2. doi: 10.1002/anie.201208294. Epub 2013 Jan 11.
Angew Chem Int Ed Engl. 2013.
PMID: 23315953
No abstract available.
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Zwitterionic uracil derivatives as potent GnRH receptor antagonists with improved pharmaceutical properties.
Regan CF, Guo Z, Chen Y, Huang CQ, Chen M, Jiang W, Rueter JK, Coon T, Chen C, Saunders J, Brown MS, Betz SF, Struthers RS, Yang C, Wen J, Madan A, Zhu YF.
Regan CF, et al.
Bioorg Med Chem Lett. 2008 Aug 15;18(16):4503-7. doi: 10.1016/j.bmcl.2008.07.059. Epub 2008 Jul 17.
Bioorg Med Chem Lett. 2008.
PMID: 18667310
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