Synthesis, stability, antiviral activity, and protease-bound structures of substrate-mimicking constrained macrocyclic inhibitors of HIV-1 protease.
Tyndall JD, Reid RC, Tyssen DP, Jardine DK, Todd B, Passmore M, March DR, Pattenden LK, Bergman DA, Alewood D, Hu SH, Alewood PF, Birch CJ, Martin JL, Fairlie DP.
Tyndall JD, et al. Among authors: alewood d, alewood pf.
J Med Chem. 2000 Sep 21;43(19):3495-504. doi: 10.1021/jm000013n.
J Med Chem. 2000.
PMID: 11000004