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Allosteric Indole Amide Inhibitors of p97: Identification of a Novel Probe of the Ubiquitin Pathway.
ACS Med Chem Lett. 2015 Dec 22;7(2):182-7. doi: 10.1021/acsmedchemlett.5b00396. eCollection 2016 Feb 11.
ACS Med Chem Lett. 2015.
PMID: 26985295
Free PMC article.
Development of highly potent and selective diaminothiazole inhibitors of cyclin-dependent kinases.
Schonbrunn E, Betzi S, Alam R, Martin MP, Becker A, Han H, Francis R, Chakrasali R, Jakkaraj S, Kazi A, Sebti SM, Cubitt CL, Gebhard AW, Hazlehurst LA, Tash JS, Georg GI.
Schonbrunn E, et al. Among authors: chakrasali r.
J Med Chem. 2013 May 23;56(10):3768-82. doi: 10.1021/jm301234k. Epub 2013 May 6.
J Med Chem. 2013.
PMID: 23600925
Free PMC article.
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Gamendazole, an orally active indazole carboxylic acid male contraceptive agent, targets HSP90AB1 (HSP90BETA) and EEF1A1 (eEF1A), and stimulates Il1a transcription in rat Sertoli cells.
Tash JS, Chakrasali R, Jakkaraj SR, Hughes J, Smith SK, Hornbaker K, Heckert LL, Ozturk SB, Hadden MK, Kinzy TG, Blagg BS, Georg GI.
Tash JS, et al. Among authors: chakrasali r.
Biol Reprod. 2008 Jun;78(6):1139-52. doi: 10.1095/biolreprod.107.062679. Epub 2008 Jan 23.
Biol Reprod. 2008.
PMID: 18218611
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A novel potent indazole carboxylic acid derivative blocks spermatogenesis and is contraceptive in rats after a single oral dose.
Tash JS, Attardi B, Hild SA, Chakrasali R, Jakkaraj SR, Georg GI.
Tash JS, et al. Among authors: chakrasali r.
Biol Reprod. 2008 Jun;78(6):1127-38. doi: 10.1095/biolreprod.106.057810. Epub 2008 Jan 23.
Biol Reprod. 2008.
PMID: 18218612
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Total synthesis and evaluation of C26-hydroxyepothilone D derivatives for photoaffinity labeling of beta-tubulin.
Reiff EA, Nair SK, Henri JT, Greiner JF, Reddy BS, Chakrasali R, David SA, Chiu TL, Amin EA, Himes RH, Vander Velde DG, Georg GI.
Reiff EA, et al. Among authors: chakrasali r.
J Org Chem. 2010 Jan 1;75(1):86-94. doi: 10.1021/jo901752v.
J Org Chem. 2010.
PMID: 19954175
Free PMC article.
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Discovery of isoxazolyl-based inhibitors of Plasmodium falciparum cGMP-dependent protein kinase.
Mahmood SU, Cheng H, Tummalapalli SR, Chakrasali R, Yadav Bheemanaboina RR, Kreiss T, Chojnowski A, Eck T, Siekierka JJ, Rotella DP.
Mahmood SU, et al. Among authors: chakrasali r.
RSC Med Chem. 2019 Dec 16;11(1):98-101. doi: 10.1039/c9md00511k. eCollection 2020 Jan 1.
RSC Med Chem. 2019.
PMID: 33479608
Free PMC article.
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Characterization of Competitive Inhibitors of Plasmodium falciparum cGMP-Dependent Protein Kinase.
Eck T, Laureano de Souza M, Delvillar M, Ashraf K, Yadav Bheemanaboina RR, Chakrasali R, Kreiss T, Siekierka JJ, Rotella DP, Bhanot P, Goodey NM.
Eck T, et al. Among authors: chakrasali r.
Chembiochem. 2022 Apr 5;23(7):e202100704. doi: 10.1002/cbic.202100704. Epub 2022 Feb 23.
Chembiochem. 2022.
PMID: 35044710
Free PMC article.
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