Akagi Y - Search Results

1

Synthetic studies of (23S,25R)-1α,25-dihydroxyvitamin D₃ 26,23-lactone (calcitriol lactone) and its derivatives.

Akagi Y, Nagata A, Odagi M, Nagasawa K. Akagi Y, et al. J Steroid Biochem Mol Biol. 2018 Mar;177:240-246. doi: 10.1016/j.jsbmb.2017.07.017. Epub 2017 Jul 27. J Steroid Biochem Mol Biol. 2018. PMID: 28757443 Review.

2

A-Ring Synthons of 19-Nor Type Vitamin D Derivatives.

Akagi Y, Yasui K, Nagasawa K. Akagi Y, et al. J Steroid Biochem Mol Biol. 2017 Oct;173:64-68. doi: 10.1016/j.jsbmb.2016.07.003. Epub 2016 Jul 18. J Steroid Biochem Mol Biol. 2017. PMID: 27436062 Review.

3

Stereoselective Synthesis of Four Calcitriol Lactone Diastereomers at C23 and C25.

Nagata A, Akagi Y, Masoud SS, Yamanaka M, Kittaka A, Uesugi M, Odagi M, Nagasawa K. Nagata A, et al. Among authors: akagi y. J Org Chem. 2019 Jun 21;84(12):7630-7641. doi: 10.1021/acs.joc.9b00403. Epub 2019 Apr 24. J Org Chem. 2019. PMID: 30985122

4

Synthesis of 24,24-Difluoro-1,3-cis-25-dihydroxy-19-norvitamin D3 Derivatives and Evaluation of Their Vitamin D Receptor-Binding Affinity.

Biswas T, Akagi Y, Usuda K, Yasui K, Shimizu I, Okamoto M, Uesugi M, Hosokawa S, Nagasawa K. Biswas T, et al. Among authors: akagi y. Biol Pharm Bull. 2016;39(8):1387-91. doi: 10.1248/bpb.b16-00316. Biol Pharm Bull. 2016. PMID: 27476947 Free article.

5

Synthesis of Diastereomers of 1,3-cis-25-Dihydroxy-19-norvitamin D3.

Usuda K, Biswas T, Yamaguchi T, Akagi Y, Yasui K, Uesugi M, Shimizu I, Hosokawa S, Nagasawa K. Usuda K, et al. Among authors: akagi y. Chem Pharm Bull (Tokyo). 2016;64(8):1190-5. doi: 10.1248/cpb.c16-00311. Chem Pharm Bull (Tokyo). 2016. PMID: 27477659 Free article.

6

Synthetic Chemical Probes That Dissect Vitamin D Activities.

Nagata A, Akagi Y, Asano L, Kotake K, Kawagoe F, Mendoza A, Masoud SS, Usuda K, Yasui K, Takemoto Y, Kittaka A, Nagasawa K, Uesugi M. Nagata A, et al. Among authors: akagi y. ACS Chem Biol. 2019 Dec 20;14(12):2851-2858. doi: 10.1021/acschembio.9b00718. Epub 2019 Oct 28. ACS Chem Biol. 2019. PMID: 31618573 Free article.

7

Discovery of a Vitamin D Receptor-Silent Vitamin D Derivative That Impairs Sterol Regulatory Element-Binding Protein In Vivo.

Kawagoe F, Mendoza A, Hayata Y, Asano L, Kotake K, Mototani S, Kawamura S, Kurosaki S, Akagi Y, Takemoto Y, Nagasawa K, Nakagawa H, Uesugi M, Kittaka A. Kawagoe F, et al. Among authors: akagi y. J Med Chem. 2021 May 13;64(9):5689-5709. doi: 10.1021/acs.jmedchem.0c02179. Epub 2021 Apr 24. J Med Chem. 2021. PMID: 33899473

8

Orally bioavailable HCV NS5A inhibitors of unsymmetrical structural class.

Nakamura H, Fujioka S, Terui T, Okuda S, Kondo K, Tamatani Y, Akagi Y, Komoda Y, Kinoshita W, Ito S, Maeda K, Ukaji Y, Inaba T. Nakamura H, et al. Among authors: akagi y. Bioorg Med Chem Lett. 2020 Sep 1;30(17):127361. doi: 10.1016/j.bmcl.2020.127361. Epub 2020 Jun 20. Bioorg Med Chem Lett. 2020. PMID: 32738974

9

Discovery of a novel unsymmetrical structural class of HCV NS5A inhibitors with low picomolar antiviral activity.

Nakamura H, Akagi Y, Terui T, Fujioka S, Komoda Y, Kinoshita W, Maeda K, Ukaji Y, Inaba T. Nakamura H, et al. Among authors: akagi y. Bioorg Med Chem Lett. 2020 Mar 1;30(5):126932. doi: 10.1016/j.bmcl.2019.126932. Epub 2019 Dec 30. Bioorg Med Chem Lett. 2020. PMID: 31952964

10

Palladium-Catalyzed β-Arylation of Cyclic α,β-Unsaturated O-Methyl Oximes with Aryl Iodides.

Akagi Y, Fukuyama S, Komatsu T. Akagi Y, et al. Chem Pharm Bull (Tokyo). 2020;68(3):288-291. doi: 10.1248/cpb.c19-01012. Chem Pharm Bull (Tokyo). 2020. PMID: 32115536 Free article.

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