Kruse CG - Search Results

1

2-Phenylpyrroles as conformationally restricted benzamide analogues. A new class of potential antipsychotics. 1.

van Wijngaarden I, Kruse CG, van Hes R, van der Heyden JA, Tulp MT. van Wijngaarden I, et al. Among authors: kruse cg. J Med Chem. 1987 Nov;30(11):2099-104. doi: 10.1021/jm00394a028. J Med Chem. 1987. PMID: 2889830

2

SLV310, a novel, potential antipsychotic, combining potent dopamine D2 receptor antagonism with serotonin reuptake inhibition.

van Hes R, Smid P, Stroomer CN, Tipker K, Tulp MT, van der Heyden JA, McCreary AC, Hesselink MB, Kruse CG. van Hes R, et al. Among authors: kruse cg. Bioorg Med Chem Lett. 2003 Feb 10;13(3):405-8. doi: 10.1016/s0960-894x(02)00996-4. Bioorg Med Chem Lett. 2003. PMID: 12565939

3

Synthesis, structure-activity relationships, and biological properties of 1-heteroaryl-4-[omega-(1H-indol-3-yl)alkyl]piperazines, novel potential antipsychotics combining potent dopamine D2 receptor antagonism with potent serotonin reuptake inhibition.

Smid P, Coolen HK, Keizer HG, van Hes R, de Moes JP, den Hartog AP, Stork B, Plekkenpol RH, Niemann LC, Stroomer CN, Tulp MT, van Stuivenberg HH, McCreary AC, Hesselink MB, Herremans AH, Kruse CG. Smid P, et al. Among authors: kruse cg. J Med Chem. 2005 Nov 3;48(22):6855-69. doi: 10.1021/jm050148z. J Med Chem. 2005. PMID: 16250644

4

Synthesis and structure-activity data of some new epibatidine analogues.

Seerden JP, Tulp MT, Scheeren HW, Kruse CG. Seerden JP, et al. Among authors: kruse cg. Bioorg Med Chem. 1998 Nov;6(11):2103-10. doi: 10.1016/s0968-0896(98)00163-1. Bioorg Med Chem. 1998. PMID: 9881100

5

New 1-aryl-4-(biarylmethylene)piperazines as potential atypical antipsychotics sharing dopamine D(2)-receptor and serotonin 5-HT(1A)-receptor affinities.

Feenstra RW, de Moes J, Hofma JJ, Kling H, Kuipers W, Long SK, Tulp MT, van der Heyden JA, Kruse CG. Feenstra RW, et al. Among authors: kruse cg. Bioorg Med Chem Lett. 2001 Sep 3;11(17):2345-9. doi: 10.1016/s0960-894x(01)00425-5. Bioorg Med Chem Lett. 2001. PMID: 11527728

6

2-Phenylpyrroles as conformationally restricted benzamide analogues. A new class of potential antipsychotics. 2.

van Wijngaarden I, Kruse CG, van der Heyden JA, Tulp MT. van Wijngaarden I, et al. Among authors: kruse cg. J Med Chem. 1988 Oct;31(10):1934-40. doi: 10.1021/jm00118a011. J Med Chem. 1988. PMID: 2902226

7

N4-unsubstituted N1-arylpiperazines as high-affinity 5-HT1A receptor ligands.

Kuipers W, van Wijngaarden I, Kruse CG, ter Horst-van Amstel M, Tulp MT, IJzerman AP. Kuipers W, et al. Among authors: kruse cg. J Med Chem. 1995 May 26;38(11):1942-54. doi: 10.1021/jm00011a014. J Med Chem. 1995. PMID: 7783126

8

5-HT1A-versus D2-receptor selectivity of flesinoxan and analogous N4-substituted N1-arylpiperazines.

Kuipers W, Kruse CG, van Wijngaarden I, Standaar PJ, Tulp MT, Veldman N, Spek AL, IJzerman AP. Kuipers W, et al. Among authors: kruse cg. J Med Chem. 1997 Jan 31;40(3):300-12. doi: 10.1021/jm960496o. J Med Chem. 1997. PMID: 9022796

9

Synthesis, biological properties, and molecular modeling investigations of novel 3,4-diarylpyrazolines as potent and selective CB(1) cannabinoid receptor antagonists.

Lange JH, Coolen HK, van Stuivenberg HH, Dijksman JA, Herremans AH, Ronken E, Keizer HG, Tipker K, McCreary AC, Veerman W, Wals HC, Stork B, Verveer PC, den Hartog AP, de Jong NM, Adolfs TJ, Hoogendoorn J, Kruse CG. Lange JH, et al. Among authors: kruse cg. J Med Chem. 2004 Jan 29;47(3):627-43. doi: 10.1021/jm031019q. J Med Chem. 2004. PMID: 14736243

10

Bioisosteric replacements of the pyrazole moiety of rimonabant: synthesis, biological properties, and molecular modeling investigations of thiazoles, triazoles, and imidazoles as potent and selective CB1 cannabinoid receptor antagonists.

Lange JH, van Stuivenberg HH, Coolen HK, Adolfs TJ, McCreary AC, Keizer HG, Wals HC, Veerman W, Borst AJ, de Looff W, Verveer PC, Kruse CG. Lange JH, et al. Among authors: kruse cg. J Med Chem. 2005 Mar 24;48(6):1823-38. doi: 10.1021/jm040843r. J Med Chem. 2005. PMID: 15771428

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