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Evolution of PI3Kγ and δ Inhibitors for Inflammatory and Autoimmune Diseases.
J Med Chem. 2019 May 23;62(10):4783-4814. doi: 10.1021/acs.jmedchem.8b01298. Epub 2018 Dec 24.
J Med Chem. 2019.
PMID: 30582813
Review.
Discovery of Highly Isoform Selective Orally Bioavailable Phosphoinositide 3-Kinase (PI3K)-γ Inhibitors.
Pemberton N, Mogemark M, Arlbrandt S, Bold P, Cox RJ, Gardelli C, Holden NS, Karabelas K, Karlsson J, Lever S, Li X, Lindmark H, Norberg M, Perry MWD, Petersen J, Rodrigo Blomqvist S, Thomas M, Tyrchan C, Westin Eriksson A, Zlatoidsky P, Öster L.
Pemberton N, et al. Among authors: westin eriksson a.
J Med Chem. 2018 Jun 28;61(12):5435-5441. doi: 10.1021/acs.jmedchem.8b00447. Epub 2018 Jun 18.
J Med Chem. 2018.
PMID: 29852070
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Discovery of AZD8154, a Dual PI3Kγδ Inhibitor for the Treatment of Asthma.
Perry MWD, Björhall K, Bold P, Brűlls M, Börjesson U, Carlsson J, Chang HA, Chen Y, Eriksson A, Fihn BM, Fransson R, Fredlund L, Ge H, Huang H, Karabelas K, Lamm Bergström E, Lever S, Lindmark H, Mogemark M, Nikitidis A, Palmgren AP, Pemberton N, Petersen J, Rodrigo Blomqvist M, Smith RW, Thomas MJ, Ullah V, Tyrchan C, Wennberg T, Westin Eriksson A, Yang W, Zhao S, Öster L.
Perry MWD, et al. Among authors: westin eriksson a.
J Med Chem. 2021 Jun 24;64(12):8053-8075. doi: 10.1021/acs.jmedchem.1c00434. Epub 2021 Jun 3.
J Med Chem. 2021.
PMID: 34080862
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Discovery and Early Clinical Development of an Inhibitor of 5-Lipoxygenase Activating Protein (AZD5718) for Treatment of Coronary Artery Disease.
Pettersen D, Broddefalk J, Emtenäs H, Hayes MA, Lemurell M, Swanson M, Ulander J, Whatling C, Amilon C, Ericsson H, Westin Eriksson A, Granberg K, Plowright AT, Shamovsky I, Dellsèn A, Sundqvist M, Någård M, Lindstedt EL.
Pettersen D, et al. Among authors: westin eriksson a.
J Med Chem. 2019 May 9;62(9):4312-4324. doi: 10.1021/acs.jmedchem.8b02004. Epub 2019 Mar 26.
J Med Chem. 2019.
PMID: 30869888
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Novel Chemical Series of 5-Lipoxygenase-Activating Protein Inhibitors for Treatment of Coronary Artery Disease.
Lemurell M, Ulander J, Emtenäs H, Winiwarter S, Broddefalk J, Swanson M, Hayes MA, Prieto Garcia L, Westin Eriksson A, Meuller J, Cassel J, Saarinen G, Yuan ZQ, Löfberg C, Karlsson S, Sundqvist M, Whatling C.
Lemurell M, et al. Among authors: westin eriksson a.
J Med Chem. 2019 May 9;62(9):4325-4349. doi: 10.1021/acs.jmedchem.8b02012. Epub 2019 Apr 15.
J Med Chem. 2019.
PMID: 30929436
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Effect of broad-spectrum matrix metalloproteinase inhibition on atherosclerotic plaque stability.
Johnson JL, Fritsche-Danielson R, Behrendt M, Westin-Eriksson A, Wennbo H, Herslof M, Elebring M, George SJ, McPheat WL, Jackson CL.
Johnson JL, et al. Among authors: westin eriksson a.
Cardiovasc Res. 2006 Aug 1;71(3):586-95. doi: 10.1016/j.cardiores.2006.05.009. Epub 2006 May 10.
Cardiovasc Res. 2006.
PMID: 16759648
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Anti-thrombotic effect of a PAI-1 inhibitor in rats given endotoxin.
Abrahamsson T, Nerme V, Strömqvist M, Akerblom B, Legnehed A, Pettersson K, Westin Eriksson A.
Abrahamsson T, et al. Among authors: westin eriksson a.
Thromb Haemost. 1996 Jan;75(1):118-26.
Thromb Haemost. 1996.
PMID: 8713790
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