Piergentili A - Search Results

1

Chemical manipulations on the 1,4-dioxane ring of 5-HT_1A receptor agonists lead to antagonists endowed with antitumor activity in prostate cancer cells.

Del Bello F, Bonifazi A, Giorgioni G, Quaglia W, Amantini C, Morelli MB, Santoni G, Battiti FO, Vistoli G, Cilia A, Piergentili A. Del Bello F, et al. Among authors: piergentili a. Eur J Med Chem. 2019 Apr 15;168:461-473. doi: 10.1016/j.ejmech.2019.02.056. Epub 2019 Feb 25. Eur J Med Chem. 2019. PMID: 30844609

2

Synthesis and dopamine receptor affinities of 2-(4-fluoro-3- hydroxyphenyl)ethylamine and N-substituted derivatives.

Claudi F, Cardellini M, Cingolani GM, Piergentili A, Peruzzi G, Balduini W. Claudi F, et al. Among authors: piergentili a. J Med Chem. 1990 Sep;33(9):2408-12. doi: 10.1021/jm00171a014. J Med Chem. 1990. PMID: 1975274

3

Synthesis and muscarinic receptors affinity of a series of antagonist bivalent ligands.

Piergentili A, Quaglia W, Tayebati SK, Paparelli F, Malmusi L, Brasili L. Piergentili A, et al. Farmaco. 1994 Feb;49(2):83-7. Farmaco. 1994. PMID: 7516166

4

Synthesis and muscarinic properties of (1S*,3R*,5R*)-trimethyl(1-methyl-6-oxabicyclo[3.1.0]hex-3-yl)methyl ammonium iodide.

Giannella M, Piergentili A, Pigini M, Quaglia W, Rafaiani G, Tayebati SK. Giannella M, et al. Among authors: piergentili a. Chem Pharm Bull (Tokyo). 1994 Jun;42(6):1286-90. doi: 10.1248/cpb.42.1286. Chem Pharm Bull (Tokyo). 1994. PMID: 8069977

5

Structure-activity relationships in 1,4-benzodioxan-related compounds. 4. Effect of aryl and alkyl substituents at position 3 on alpha-adrenoreceptor blocking activity.

Quaglia W, Pigini M, Tayebati SK, Piergentili A, Giannella M, Marucci G, Melchiorre C. Quaglia W, et al. Among authors: piergentili a. J Med Chem. 1993 May 28;36(11):1520-8. doi: 10.1021/jm00063a002. J Med Chem. 1993. PMID: 8098772

6

Synthesis, absolute configuration, and biological profile of the enantiomers of trans-[2-(2,6-dimethoxyphenoxy)ethyl] [(3-p-tolyl-2,3-dihydro-1,4-benzodioxin-2-yl)methyl]amine (mephendioxan), a potent competitive alpha 1A-adrenoreceptor antagonist.

Quaglia W, Pigini M, Tayebati SK, Piergentili A, Giannella M, Leonardi A, Taddei C, Melchiorre C. Quaglia W, et al. Among authors: piergentili a. J Med Chem. 1996 May 24;39(11):2253-8. doi: 10.1021/jm960069a. J Med Chem. 1996. PMID: 8667368

7

Bicyclic dioxolanes as potential antimuscarinic agents.

Piergentili A, Angeli P, Giannella M, Pigini M, Quaglia W, Tayebati SK. Piergentili A, et al. Arzneimittelforschung. 1996 Feb;46(2):99-105. Arzneimittelforschung. 1996. PMID: 8720297

8

Structure-activity relationships in 1,4-benzodioxan-related compounds. 5. Effects of modification of the side chain on alpha-adrenoreceptor blocking activity.

Quaglia W, Giannella M, Marucci G, Piergentili A, Pigini M, Tayebati SK, Melchiorre C. Quaglia W, et al. Among authors: piergentili a. Farmaco. 1996 Jan;51(1):27-32. Farmaco. 1996. PMID: 8721758

9

Muscarinic thioligands with cyclopentane nucleus.

Piergentili A, Pigini M, Quaglia W, Tayebati SK, Amenta F, Sabbatini M, Giannella M. Piergentili A, et al. Bioorg Med Chem. 1996 Dec;4(12):2193-9. doi: 10.1016/s0968-0896(96)00231-3. Bioorg Med Chem. 1996. PMID: 9022982

10

Synthesis and structure-activity relationship studies in a series of 2-substituted 1,3-dioxolanes modified at the cationic head.

Angeli P, Brasili L, Cingolani ML, Marucci G, Piergentili A, Pigini M, Quaglia W. Angeli P, et al. Among authors: piergentili a. Bioorg Med Chem. 1997 Apr;5(4):731-7. doi: 10.1016/s0968-0896(97)00017-5. Bioorg Med Chem. 1997. PMID: 9158872

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