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Truncated (N)-Methanocarba Nucleosides as Partial Agonists at Mouse and Human A3 Adenosine Receptors: Affinity Enhancement by N6-(2-Phenylethyl) Substitution.
J Med Chem. 2020 Apr 23;63(8):4334-4348. doi: 10.1021/acs.jmedchem.0c00235. Epub 2020 Apr 9.
J Med Chem. 2020.
PMID: 32271569
Free PMC article.
Design and in Vivo Characterization of A1 Adenosine Receptor Agonists in the Native Ribose and Conformationally Constrained (N)-Methanocarba Series.
Tosh DK, Rao H, Bitant A, Salmaso V, Mannes P, Lieberman DI, Vaughan KL, Mattison JA, Rothwell AC, Auchampach JA, Ciancetta A, Liu N, Cui Z, Gao ZG, Reitman ML, Gavrilova O, Jacobson KA.
Tosh DK, et al. Among authors: lieberman di.
J Med Chem. 2019 Feb 14;62(3):1502-1522. doi: 10.1021/acs.jmedchem.8b01662. Epub 2019 Jan 3.
J Med Chem. 2019.
PMID: 30605331
Free PMC article.
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Structure activity relationship of 2-arylalkynyl-adenine derivatives as human A3 adenosine receptor antagonists.
Yu J, Mannes P, Jung YH, Ciancetta A, Bitant A, Lieberman DI, Khaznadar S, Auchampach JA, Gao ZG, Jacobson KA.
Yu J, et al. Among authors: lieberman di.
Medchemcomm. 2018 Oct 18;9(11):1920-1932. doi: 10.1039/c8md00317c. eCollection 2018 Nov 1.
Medchemcomm. 2018.
PMID: 30568760
Free PMC article.
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Structure-Activity Relationship of Heterocyclic P2Y14 Receptor Antagonists: Removal of the Zwitterionic Character with Piperidine Bioisosteres.
Jung YH, Salmaso V, Wen Z, Bennett JM, Phung NB, Lieberman DI, Gopinatth V, Randle JCR, Chen Z, Salvemini D, Karcz TP, Cook DN, Jacobson KA.
Jung YH, et al. Among authors: lieberman di.
J Med Chem. 2021 Apr 22;64(8):5099-5122. doi: 10.1021/acs.jmedchem.1c00164. Epub 2021 Mar 31.
J Med Chem. 2021.
PMID: 33787273
Free PMC article.
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Bridged Piperidine Analogues of a High Affinity Naphthalene-Based P2Y14R Antagonist.
Wen Z, Salmaso V, Jung YH, Phung NB, Gopinatth V, Shah Q, Patterson AT, Randle JCR, Chen Z, Salvemini D, Lieberman DI, Whitehead GS, Karcz TP, Cook DN, Jacobson KA.
Wen Z, et al. Among authors: lieberman di.
J Med Chem. 2022 Feb 24;65(4):3434-3459. doi: 10.1021/acs.jmedchem.1c01964. Epub 2022 Feb 3.
J Med Chem. 2022.
PMID: 35113556
Free PMC article.
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A3 adenosine receptor activation mechanisms: molecular dynamics analysis of inactive, active, and fully active states.
Ciancetta A, Rubio P, Lieberman DI, Jacobson KA.
Ciancetta A, et al. Among authors: lieberman di.
J Comput Aided Mol Des. 2019 Nov;33(11):983-996. doi: 10.1007/s10822-019-00246-4. Epub 2019 Nov 22.
J Comput Aided Mol Des. 2019.
PMID: 31758354
Free PMC article.
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