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5,6-Dihydroxypyrimidine Scaffold to Target HIV-1 Nucleocapsid Protein.
ACS Med Chem Lett. 2020 Mar 19;11(5):766-772. doi: 10.1021/acsmedchemlett.9b00608. eCollection 2020 May 14.
ACS Med Chem Lett. 2020.
PMID: 32435383
Free PMC article.
Structure-Based Identification of HIV-1 Nucleocapsid Protein Inhibitors Active against Wild-Type and Drug-Resistant HIV-1 Strains.
Mori M, Kovalenko L, Malancona S, Saladini F, De Forni D, Pires M, Humbert N, Real E, Botzanowski T, Cianférani S, Giannini A, Dasso Lang MC, Cugia G, Poddesu B, Lori F, Zazzi M, Harper S, Summa V, Mely Y, Botta M.
Mori M, et al. Among authors: dasso lang mc.
ACS Chem Biol. 2018 Jan 19;13(1):253-266. doi: 10.1021/acschembio.7b00907. Epub 2017 Dec 28.
ACS Chem Biol. 2018.
PMID: 29235845
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Synthesis and Evaluation of Bifunctional Aminothiazoles as Antiretrovirals Targeting the HIV-1 Nucleocapsid Protein.
Mori M, Dasso Lang MC, Saladini F, Palombi N, Kovalenko L, De Forni D, Poddesu B, Friggeri L, Giannini A, Malancona S, Summa V, Zazzi M, Mely Y, Botta M.
Mori M, et al. Among authors: dasso lang mc.
ACS Med Chem Lett. 2018 Dec 7;10(4):463-468. doi: 10.1021/acsmedchemlett.8b00506. eCollection 2019 Apr 11.
ACS Med Chem Lett. 2018.
PMID: 30996780
Free PMC article.
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Synthesis of linear and cyclic guazatine derivatives endowed with antibacterial activity.
Maccari G, Sanfilippo S, De Luca F, Deodato D, Casian A, Dasso Lang MC, Zamperini C, Dreassi E, Rossolini GM, Docquier JD, Botta M.
Maccari G, et al. Among authors: dasso lang mc.
Bioorg Med Chem Lett. 2014 Dec 1;24(23):5525-9. doi: 10.1016/j.bmcl.2014.09.081. Epub 2014 Oct 14.
Bioorg Med Chem Lett. 2014.
PMID: 25455183
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Development and in Vitro Evaluation of a Microbicide Gel Formulation for a Novel Non-Nucleoside Reverse Transcriptase Inhibitor Belonging to the N-Dihydroalkyloxybenzyloxopyrimidines (N-DABOs) Family.
Tintori C, Brai A, Dasso Lang MC, Deodato D, Greco AM, Bizzarri BM, Cascone L, Casian A, Zamperini C, Dreassi E, Crespan E, Maga G, Vanham G, Ceresola E, Canducci F, Ariën KK, Botta M.
Tintori C, et al. Among authors: dasso lang mc.
J Med Chem. 2016 Mar 24;59(6):2747-59. doi: 10.1021/acs.jmedchem.5b01979. Epub 2016 Mar 8.
J Med Chem. 2016.
PMID: 26898379
Free article.
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Insights into the interaction of high potency inhibitor IRC-083864 with phosphatase CDC25.
Sarkis M, Miteva MA, Dasso Lang MC, Jaouen M, Sari MA, Galcéra MO, Ethève-Quelquejeu M, Garbay C, Bertho G, Braud E.
Sarkis M, et al. Among authors: dasso lang mc.
Proteins. 2017 Apr;85(4):593-601. doi: 10.1002/prot.25236. Epub 2017 Jan 18.
Proteins. 2017.
PMID: 28056492
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