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Structure-activity relationship studies for the development of inhibitors of murine adipose triglyceride lipase (ATGL).
Bioorg Med Chem. 2020 Aug 15;28(16):115610. doi: 10.1016/j.bmc.2020.115610. Epub 2020 Jul 4.
Bioorg Med Chem. 2020.
PMID: 32690265
Free article.
Atglistatin ameliorates functional decline in heart failure via adipocyte-specific inhibition of adipose triglyceride lipase.
Parajuli N, Takahara S, Matsumura N, Kim TT, Ferdaoussi M, Migglautsch AK, Zechner R, Breinbauer R, Kershaw EE, Dyck JRB.
Parajuli N, et al. Among authors: migglautsch ak.
Am J Physiol Heart Circ Physiol. 2018 Oct 1;315(4):H879-H884. doi: 10.1152/ajpheart.00308.2018. Epub 2018 Jun 22.
Am J Physiol Heart Circ Physiol. 2018.
PMID: 29932770
Free article.
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Inhibition of ATGL in adipose tissue ameliorates isoproterenol-induced cardiac remodeling by reducing adipose tissue inflammation.
Takahara S, Ferdaoussi M, Srnic N, Maayah ZH, Soni S, Migglautsch AK, Breinbauer R, Kershaw EE, Dyck JRB.
Takahara S, et al. Among authors: migglautsch ak.
Am J Physiol Heart Circ Physiol. 2021 Jan 1;320(1):H432-H446. doi: 10.1152/ajpheart.00737.2020. Epub 2020 Nov 13.
Am J Physiol Heart Circ Physiol. 2021.
PMID: 33185110
Free PMC article.
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Pharmacological inhibition of adipose tissue adipose triglyceride lipase by Atglistatin prevents catecholamine-induced myocardial damage.
Thiele A, Luettges K, Ritter D, Beyhoff N, Smeir E, Grune J, Steinhoff JS, Schupp M, Klopfleisch R, Rothe M, Wilck N, Bartolomaeus H, Migglautsch AK, Breinbauer R, Kershaw EE, Grabner GF, Zechner R, Kintscher U, Foryst-Ludwig A.
Thiele A, et al. Among authors: migglautsch ak.
Cardiovasc Res. 2022 Aug 24;118(11):2488-2505. doi: 10.1093/cvr/cvab182.
Cardiovasc Res. 2022.
PMID: 34061169
Free PMC article.
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Enzymatic aerobic alkene cleavage catalyzed by a Mn(3+) -dependent proteinase a homologue.
Rajagopalan A, Schober M, Emmerstorfer A, Hammerer L, Migglautsch A, Seisser B, Glueck SM, Niehaus F, Eck J, Pichler H, Gruber K, Kroutil W.
Rajagopalan A, et al.
Chembiochem. 2013 Dec 16;14(18):2427-30. doi: 10.1002/cbic.201300601. Epub 2013 Nov 4.
Chembiochem. 2013.
PMID: 24318692
No abstract available.
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