Skip to main page content
U.S. flag

An official website of the United States government

Dot gov

The .gov means it’s official.
Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you’re on a federal government site.

Https

The site is secure.
The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.

Access keys NCBI Homepage MyNCBI Homepage Main Content Main Navigation

Search Page

Filters

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

Search Results

15 results

Filters applied: . Clear all
Results are displayed in a computed author sort order. The Results By Year timeline is not available.
Page 1
Pyrazolones as inhibitors of immune checkpoint blocking the PD-1/PD-L1 interaction.
Le Biannic R, Magnez R, Klupsch F, Leleu-Chavain N, Thiroux B, Tardy M, El Bouazzati H, Dezitter X, Renault N, Vergoten G, Bailly C, Quesnel B, Thuru X, Millet R. Le Biannic R, et al. Among authors: klupsch f. Eur J Med Chem. 2022 Jun 5;236:114343. doi: 10.1016/j.ejmech.2022.114343. Epub 2022 Apr 4. Eur J Med Chem. 2022. PMID: 35429911
4-Oxo-1,4-dihydropyridines as selective CB₂ cannabinoid receptor ligands. Part 2: discovery of new agonists endowed with protective effect against experimental colitis.
El Bakali J, Gilleron P, Body-Malapel M, Mansouri R, Muccioli GG, Djouina M, Barczyk A, Klupsch F, Andrzejak V, Lipka E, Furman C, Lambert DM, Chavatte P, Desreumaux P, Millet R. El Bakali J, et al. Among authors: klupsch f. J Med Chem. 2012 Oct 25;55(20):8948-52. doi: 10.1021/jm3008568. Epub 2012 Oct 12. J Med Chem. 2012. PMID: 23017078
One- or Two-Step Synthesis of C-8 and N-9 Substituted Purines.
Bollier M, Klupsch F, Six P, Dubuquoy L, Azaroual N, Millet R, Leleu-Chavain N. Bollier M, et al. Among authors: klupsch f. J Org Chem. 2018 Jan 5;83(1):422-430. doi: 10.1021/acs.joc.7b02269. Epub 2017 Dec 14. J Org Chem. 2018. PMID: 29192784
Synthesis and biological evaluation of ferrocene-based cannabinoid receptor 2 ligands.
Sansook S, Tuo W, Bollier M, Barczyk A, Dezitter X, Klupsch F, Leleu-Chavain N, Farce A, Tizzard GJ, Coles SJ, Spencer J, Millet R. Sansook S, et al. Among authors: klupsch f. Future Med Chem. 2018 Mar 1;10(6):631-638. doi: 10.4155/fmc-2017-0200. Epub 2018 Feb 8. Future Med Chem. 2018. PMID: 29419319 Free article.
Novel PD-L1-Targeted Phenyl-Pyrazolone Derivatives with Antioxidant Properties.
Regnault R, Klupsch F, El-Bouazzati H, Magnez R, Le Biannic R, Leleu-Chavain N, Ahouari H, Vezin H, Millet R, Goossens JF, Thuru X, Bailly C. Regnault R, et al. Among authors: klupsch f. Molecules. 2023 Apr 15;28(8):3491. doi: 10.3390/molecules28083491. Molecules. 2023. PMID: 37110727 Free PMC article.
Activity of pyridyl-pyrazolone derivatives against Trypanosoma cruzi.
Batista DDGJ, de Almeida Fiuza LF, Klupsch F, da Costa KN, Batista MM, da Conceição K, Bouafia H, Vergoten G, Millet R, Thuru X, Bailly C, Soeiro MNC. Batista DDGJ, et al. Among authors: klupsch f. Exp Parasitol. 2024 May 15:108787. doi: 10.1016/j.exppara.2024.108787. Online ahead of print. Exp Parasitol. 2024. PMID: 38759776 Free article.
New benzo[5,6]pyrrolizino[1,2-b]quinolines as cytotoxic agents.
Perzyna A, Klupsch F, Houssin R, Pommery N, Lemoine A, Hénichart JP. Perzyna A, et al. Among authors: klupsch f. Bioorg Med Chem Lett. 2004 May 3;14(9):2363-5. doi: 10.1016/j.bmcl.2004.01.097. Bioorg Med Chem Lett. 2004. PMID: 15081041
15 results