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Antimalarial Imidazopyridines Incorporating an Intramolecular Hydrogen Bonding Motif: Medicinal Chemistry and Mechanistic Studies.
ACS Infect Dis. 2023 Apr 14;9(4):928-942. doi: 10.1021/acsinfecdis.2c00584. Epub 2023 Mar 22.
ACS Infect Dis. 2023.
PMID: 36946433
Free PMC article.
Novel 3-Trifluoromethyl-1,2,4-oxadiazole Analogues of Astemizole with Multi-stage Antiplasmodium Activity and In Vivo Efficacy in a Plasmodium berghei Mouse Malaria Infection Model.
Mambwe D, Korkor CM, Mabhula A, Ngqumba Z, Cloete C, Kumar M, Barros PL, Leshabane M, Coertzen D, Taylor D, Gibhard L, Njoroge M, Lawrence N, Reader J, Moreira DR, Birkholtz LM, Wittlin S, Egan TJ, Chibale K.
Mambwe D, et al. Among authors: korkor cm.
J Med Chem. 2022 Dec 22;65(24):16695-16715. doi: 10.1021/acs.jmedchem.2c01516. Epub 2022 Dec 12.
J Med Chem. 2022.
PMID: 36507890
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Innovation Experiences from Africa-Led Drug Discovery at the Holistic Drug Discovery and Development (H3D) Centre.
Singh V, Mambwe D, Korkor CM, Chibale K.
Singh V, et al. Among authors: korkor cm.
ACS Med Chem Lett. 2022 Jul 11;13(8):1221-1230. doi: 10.1021/acsmedchemlett.2c00142. eCollection 2022 Aug 11.
ACS Med Chem Lett. 2022.
PMID: 35978699
Free PMC article.
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Antimalarial Benzimidazole Derivatives Incorporating Phenolic Mannich Base Side Chains Inhibit Microtubule and Hemozoin Formation: Structure-Activity Relationship and In Vivo Oral Efficacy Studies.
Dziwornu GA, Coertzen D, Leshabane M, Korkor CM, Cloete CK, Njoroge M, Gibhard L, Lawrence N, Reader J, van der Watt M, Wittlin S, Birkholtz LM, Chibale K.
Dziwornu GA, et al. Among authors: korkor cm.
J Med Chem. 2021 Apr 22;64(8):5198-5215. doi: 10.1021/acs.jmedchem.1c00354. Epub 2021 Apr 12.
J Med Chem. 2021.
PMID: 33844521
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Intrinsic fluorescence properties of antimalarial pyrido[1,2-a]benzimidazoles facilitate subcellular accumulation and mechanistic studies in the human malaria parasite Plasmodium falciparum.
Korkor CM, Garnie LF, Amod L, Egan TJ, Chibale K.
Korkor CM, et al.
Org Biomol Chem. 2020 Nov 4;18(42):8668-8676. doi: 10.1039/d0ob01730b.
Org Biomol Chem. 2020.
PMID: 33078179
Free PMC article.
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