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Discovery and Optimization of a Novel Macrocyclic Amidinourea Series Active as Acidic Mammalian Chitinase Inhibitors.
ACS Med Chem Lett. 2023 Mar 21;14(4):417-424. doi: 10.1021/acsmedchemlett.2c00472. eCollection 2023 Apr 13.
ACS Med Chem Lett. 2023.
PMID: 37077400
Free PMC article.
Focused library of phenyl-fused macrocyclic amidinoureas as antifungal agents.
Balestri LJI, D'Agostino I, Rango E, Vagaggini C, Marchitiello R, Mariotti M, Casian A, Deodato D, Truglio GI, Orofino F, Sanguinetti M, Bugli F, Botta L, Dreassi E.
Balestri LJI, et al.
Mol Divers. 2022 Dec;26(6):3399-3409. doi: 10.1007/s11030-022-10388-7. Epub 2022 Feb 10.
Mol Divers. 2022.
PMID: 35143033
Free PMC article.
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