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Discovery and Optimization of a Novel Macrocyclic Amidinourea Series Active as Acidic Mammalian Chitinase Inhibitors.
ACS Med Chem Lett. 2023 Mar 21;14(4):417-424. doi: 10.1021/acsmedchemlett.2c00472. eCollection 2023 Apr 13.
ACS Med Chem Lett. 2023.
PMID: 37077400
Free PMC article.
Design and synthesis of a novel inhibitor of T. Viride chitinase through an in silico target fishing protocol.
Maccari G, Deodato D, Fiorucci D, Orofino F, Truglio GI, Pasero C, Martini R, De Luca F, Docquier JD, Botta M.
Maccari G, et al. Among authors: truglio gi.
Bioorg Med Chem Lett. 2017 Aug 1;27(15):3332-3336. doi: 10.1016/j.bmcl.2017.06.016. Epub 2017 Jun 10.
Bioorg Med Chem Lett. 2017.
PMID: 28610983
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Alkyl-guanidine Compounds as Potent Broad-Spectrum Antibacterial Agents: Chemical Library Extension and Biological Characterization.
Pasero C, D'Agostino I, De Luca F, Zamperini C, Deodato D, Truglio GI, Sannio F, Del Prete R, Ferraro T, Visaggio D, Mancini A, Guglielmi MB, Visca P, Docquier JD, Botta M.
Pasero C, et al. Among authors: truglio gi.
J Med Chem. 2018 Oct 25;61(20):9162-9176. doi: 10.1021/acs.jmedchem.8b00619. Epub 2018 Oct 11.
J Med Chem. 2018.
PMID: 30265809
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In vitro characterization, ADME analysis, and histological and toxicological evaluation of BM1, a macrocyclic amidinourea active against azole-resistant Candida strains.
Orofino F, Truglio GI, Fiorucci D, D'Agostino I, Borgini M, Poggialini F, Zamperini C, Dreassi E, Maccari L, Torelli R, Martini C, Bernabei M, Meis JF, Khandelwal NK, Prasad R, Sanguinetti M, Bugli F, Botta M.
Orofino F, et al. Among authors: truglio gi.
Int J Antimicrob Agents. 2020 Mar;55(3):105865. doi: 10.1016/j.ijantimicag.2019.105865. Epub 2019 Dec 20.
Int J Antimicrob Agents. 2020.
PMID: 31866465
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Focused library of phenyl-fused macrocyclic amidinoureas as antifungal agents.
Balestri LJI, D'Agostino I, Rango E, Vagaggini C, Marchitiello R, Mariotti M, Casian A, Deodato D, Truglio GI, Orofino F, Sanguinetti M, Bugli F, Botta L, Dreassi E.
Balestri LJI, et al. Among authors: truglio gi.
Mol Divers. 2022 Dec;26(6):3399-3409. doi: 10.1007/s11030-022-10388-7. Epub 2022 Feb 10.
Mol Divers. 2022.
PMID: 35143033
Free PMC article.
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CanB, a Druggable Cellular Target in Mycobacterium tuberculosis.
Degiacomi G, Gianibbi B, Recchia D, Stelitano G, Truglio GI, Marra P, Stamilla A, Makarov V, Chiarelli LR, Manetti F, Pasca MR.
Degiacomi G, et al. Among authors: truglio gi.
ACS Omega. 2023 Jul 3;8(28):25209-25220. doi: 10.1021/acsomega.3c02311. eCollection 2023 Jul 18.
ACS Omega. 2023.
PMID: 37483251
Free PMC article.
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