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Development of submicromolar 17β-HSD10 inhibitors and their in vitro and in vivo evaluation.
Eur J Med Chem. 2023 Oct 5;258:115593. doi: 10.1016/j.ejmech.2023.115593. Epub 2023 Jun 24.
Eur J Med Chem. 2023.
PMID: 37390508
1-(Benzo[d]thiazol-2-yl)-3-phenylureas as dual inhibitors of casein kinase 1 and ABAD enzymes for treatment of neurodegenerative disorders.
Benek O, Hroch L, Aitken L, Gunn-Moore F, Vinklarova L, Kuca K, Perez DI, Perez C, Martinez A, Fisar Z, Musilek K.
Benek O, et al. Among authors: vinklarova l.
J Enzyme Inhib Med Chem. 2018 Dec;33(1):665-670. doi: 10.1080/14756366.2018.1445736.
J Enzyme Inhib Med Chem. 2018.
PMID: 29536773
Free PMC article.
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Novel Benzothiazole-based Ureas as 17β-HSD10 Inhibitors, A Potential Alzheimer's Disease Treatment.
Aitken L, Benek O, McKelvie BE, Hughes RE, Hroch L, Schmidt M, Major LL, Vinklarova L, Kuca K, Smith TK, Musilek K, Gunn-Moore FJ.
Aitken L, et al. Among authors: vinklarova l.
Molecules. 2019 Jul 29;24(15):2757. doi: 10.3390/molecules24152757.
Molecules. 2019.
PMID: 31362457
Free PMC article.
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Benzothiazolyl Ureas are Low Micromolar and Uncompetitive Inhibitors of 17β-HSD10 with Implications to Alzheimer's Disease Treatment.
Schmidt M, Benek O, Vinklarova L, Hrabinova M, Zemanova L, Chribek M, Kralova V, Hroch L, Dolezal R, Lycka A, Prchal L, Jun D, Aitken L, Gunn-Moore F, Kuca K, Musilek K.
Schmidt M, et al. Among authors: vinklarova l.
Int J Mol Sci. 2020 Mar 17;21(6):2059. doi: 10.3390/ijms21062059.
Int J Mol Sci. 2020.
PMID: 32192199
Free PMC article.
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Friend or enemy? Review of 17β-HSD10 and its role in human health or disease.
Vinklarova L, Schmidt M, Benek O, Kuca K, Gunn-Moore F, Musilek K.
Vinklarova L, et al.
J Neurochem. 2020 Nov;155(3):231-249. doi: 10.1111/jnc.15027. Epub 2020 May 23.
J Neurochem. 2020.
PMID: 32306391
Free article.
Review.
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Effects of novel 17β-hydroxysteroid dehydrogenase type 10 inhibitors on mitochondrial respiration.
Fišar Z, Musílek K, Benek O, Hroch L, Vinklářová L, Schmidt M, Hroudová J, Raboch J.
Fišar Z, et al. Among authors: vinklarova l.
Toxicol Lett. 2021 Mar 15;339:12-19. doi: 10.1016/j.toxlet.2020.12.012. Epub 2020 Dec 24.
Toxicol Lett. 2021.
PMID: 33359020
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