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Activation and Signaling Mechanism Revealed by Cannabinoid Receptor-Gi Complex Structures.
Cell. 2020 Feb 20;180(4):655-665.e18. doi: 10.1016/j.cell.2020.01.008. Epub 2020 Jan 30.
Cell. 2020.
PMID: 32004463
Free PMC article.
Novel Functionalized Cannabinoid Receptor Probes: Development of Exceptionally Potent Agonists.
Jiang S, Iliopoulos-Tsoutsouvas C, Tong F, Brust CA, Keenan CM, Raghav JG, Hua T, Wu S, Ho JH, Wu Y, Grim TW, Zvonok N, Thakur GA, Liu ZJ, Sharkey KA, Bohn LM, Nikas SP, Makriyannis A.
Jiang S, et al. Among authors: brust ca.
J Med Chem. 2021 Apr 8;64(7):3870-3884. doi: 10.1021/acs.jmedchem.0c02053. Epub 2021 Mar 24.
J Med Chem. 2021.
PMID: 33761251
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Improved cyclobutyl nabilone analogs as potent CB1 receptor agonists.
Papanastasiou IP, Georgiadis MO, Iliopoulos-Tsoutsouvas C, Paronis CA, Brust CA, Tran NK, Ji L, Ma X, Wood JT, Zvonok N, Tong F, Bohn LM, Nikas SP, Makriyannis A.
Papanastasiou IP, et al. Among authors: brust ca.
Eur J Med Chem. 2022 Feb 15;230:114027. doi: 10.1016/j.ejmech.2021.114027. Epub 2021 Dec 27.
Eur J Med Chem. 2022.
PMID: 35051750
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Structural and functional insights into the G protein-coupled receptors: CB1 and CB2.
Brust CA, Swanson MA, Bohn LM.
Brust CA, et al.
Biochem Soc Trans. 2023 Aug 31;51(4):1533-1543. doi: 10.1042/BST20221316.
Biochem Soc Trans. 2023.
PMID: 37646476
Free PMC article.
Review.
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