Burgess JP - Search Results

1

Conformationally constrained analogues of N-(piperidinyl)-5-(4-chlorophenyl)-1-(2,4- dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide (SR141716): design, synthesis, computational analysis, and biological evaluations.

Zhang Y, Burgess JP, Brackeen M, Gilliam A, Mascarella SW, Page K, Seltzman HH, Thomas BF. Zhang Y, et al. Among authors: burgess jp. J Med Chem. 2008 Jun 26;51(12):3526-39. doi: 10.1021/jm8000778. J Med Chem. 2008. PMID: 18512901

2

Discovery of an opioid kappa receptor selective pure antagonist from a library of N-substituted 4beta-methyl-5-(3-hydroxyphenyl)morphans.

Thomas JB, Atkinson RN, Namdev N, Rothman RB, Gigstad KM, Fix SE, Mascarella SW, Burgess JP, Vinson NA, Xu H, Dersch CM, Cantrell BE, Zimmerman DM, Carroll FI. Thomas JB, et al. Among authors: burgess jp. J Med Chem. 2002 Aug 1;45(16):3524-30. doi: 10.1021/jm020084h. J Med Chem. 2002. PMID: 12139463

3

Complete 1H and 13C assignments of fluorinated analogs of dehydroepiandrosterone.

Burgess JP, Wintermute JS, Thomas BF, Kapetanovic IM. Burgess JP, et al. Magn Reson Chem. 2006 Nov;44(11):1051-3. doi: 10.1002/mrc.1874. Magn Reson Chem. 2006. PMID: 16835888

4

Synthesis and transporter binding properties of 2,3-diphenyltropane stereoisomers. Comparison to 3beta-phenyltropane-2beta-carboxylic acid esters.

Chang AC, Burgess JP, Mascarella SW, Abraham P, Kuhar MJ, Carroll FI. Chang AC, et al. Among authors: burgess jp. J Med Chem. 1997 Apr 11;40(8):1247-51. doi: 10.1021/jm960703k. J Med Chem. 1997. PMID: 9111298

5

N-substituted octahydro-4a-(3-hydroxyphenyl)-10a-methyl-benzo[g]isoquinolines are opioid receptor pure antagonists.

Thomas JB, Mascarella SW, Burgess JP, Xu H, McCullough KB, Rothman RB, Flippen-Anderson JL, George CF, Cantrell BE, Zimmerman DM, Carroll FI. Thomas JB, et al. Among authors: burgess jp. Bioorg Med Chem Lett. 1998 Nov 17;8(22):3149-52. doi: 10.1016/s0960-894x(98)00576-9. Bioorg Med Chem Lett. 1998. PMID: 9873693

6

(+/-)-4-[(N-allyl-cis-3-methyl-4-piperidinyl)phenylamino]-N,N-diethylbenzamide displays selective binding for the delta opioid receptor.

Thomas JB, Herault XM, Rothman RB, Burgess JP, Mascarella SW, Xu H, Horel RB, Dersch CM, Carroll FI. Thomas JB, et al. Among authors: burgess jp. Bioorg Med Chem Lett. 1999 Oct 18;9(20):3053-6. doi: 10.1016/s0960-894x(99)00525-9. Bioorg Med Chem Lett. 1999. PMID: 10571174

7

4-[(8-Alkyl-8-azabicyclo[3.2.1]octyl-3-yl)-3-arylanilino]-N,N-diethylbenzamides: high affinity, selective ligands for the delta opioid receptor illustrate factors important to antagonist activity.

Thomas JB, Atkinson RN, Rothman RB, Burgess JP, Mascarella SW, Dersch CM, Xu H, Carroll FI. Thomas JB, et al. Among authors: burgess jp. Bioorg Med Chem Lett. 2000 Jun 5;10(11):1281-4. doi: 10.1016/s0960-894x(00)00209-2. Bioorg Med Chem Lett. 2000. PMID: 10866400

8

Factors influencing agonist potency and selectivity for the opioid delta receptor are revealed in structure-activity relationship studies of the 4-[(N-substituted-4-piperidinyl)arylamino]-N,N-diethylbenzamides.

Thomas JB, Herault XM, Rothman RB, Atkinson RN, Burgess JP, Mascarella SW, Dersch CM, Xu H, Flippen-Anderson JL, George CF, Carroll FI. Thomas JB, et al. Among authors: burgess jp. J Med Chem. 2001 Mar 15;44(6):972-87. doi: 10.1021/jm000427g. J Med Chem. 2001. PMID: 11300879

9

Identification of [14C]fluasterone metabolites in urine and feces collected from dogs after subcutaneous and oral administration of [14C]fluasterone.

Burgess JP, Green JS, Hill JM, Zhan Q, Lindeblad M, Lyubimov A, Kapetanovic IM, Schwartz A, Thomas BF. Burgess JP, et al. Drug Metab Dispos. 2009 May;37(5):1089-97. doi: 10.1124/dmd.108.023614. Epub 2009 Feb 5. Drug Metab Dispos. 2009. PMID: 19196848 Free PMC article.

10

Caged Naloxone: Synthesis, Characterization, and Stability of 3- O-(4,5-Dimethoxy-2-nitrophenyl)carboxymethyl Naloxone (CNV-NLX).

Lewin AH, Fix SE, Zhong D, Mayer LD, Burgess JP, Mascarella SW, Reddy PA, Seltzman HH, Carroll FI. Lewin AH, et al. Among authors: burgess jp. ACS Chem Neurosci. 2018 Mar 21;9(3):563-567. doi: 10.1021/acschemneuro.7b00378. Epub 2017 Dec 8. ACS Chem Neurosci. 2018. PMID: 29154536

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