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Open-source discovery of chemical leads for next-generation chemoprotective antimalarials.
Science. 2018 Dec 7;362(6419):eaat9446. doi: 10.1126/science.aat9446.
Science. 2018.
PMID: 30523084
Free PMC article.
Probing the Open Global Health Chemical Diversity Library for Multistage-Active Starting Points for Next-Generation Antimalarials.
Abraham M, Gagaring K, Martino ML, Vanaerschot M, Plouffe DM, Calla J, Godinez-Macias KP, Du AY, Wree M, Antonova-Koch Y, Eribez K, Luth MR, Ottilie S, Fidock DA, McNamara CW, Winzeler EA.
Abraham M, et al. Among authors: eribez k.
ACS Infect Dis. 2020 Apr 10;6(4):613-628. doi: 10.1021/acsinfecdis.9b00482. Epub 2020 Mar 4.
ACS Infect Dis. 2020.
PMID: 32078764
Free PMC article.
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Investigation of the in vitro and in vivo efficacy of peptoid-based HDAC inhibitors with dual-stage antiplasmodial activity.
Mackwitz MKW, Hesping E, Eribez K, Schöler A, Antonova-Koch Y, Held J, Winzeler EA, Andrews KT, Hansen FK.
Mackwitz MKW, et al. Among authors: eribez k.
Eur J Med Chem. 2021 Feb 5;211:113065. doi: 10.1016/j.ejmech.2020.113065. Epub 2020 Dec 5.
Eur J Med Chem. 2021.
PMID: 33360801
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Synthesis and Structure-Activity Relationship of Dual-Stage Antimalarial Pyrazolo[3,4-b]pyridines.
Eagon S, Hammill JT, Sigal M, Ahn KJ, Tryhorn JE, Koch G, Belanger B, Chaplan CA, Loop L, Kashtanova AS, Yniguez K, Lazaro H, Wilkinson SP, Rice AL, Falade MO, Takahashi R, Kim K, Cheung A, DiBernardo C, Kimball JJ, Winzeler EA, Eribez K, Mittal N, Gamo FJ, Crespo B, Churchyard A, García-Barbazán I, Baum J, Anderson MO, Laleu B, Guy RK.
Eagon S, et al. Among authors: eribez k.
J Med Chem. 2020 Oct 22;63(20):11902-11919. doi: 10.1021/acs.jmedchem.0c01152. Epub 2020 Oct 1.
J Med Chem. 2020.
PMID: 32945666
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Optimal 10-Aminoartemisinins With Potent Transmission-Blocking Capabilities for New Artemisinin Combination Therapies-Activities Against Blood Stage P. falciparum Including PfKI3 C580Y Mutants and Liver Stage P. berghei Parasites.
Wong HN, Padín-Irizarry V, van der Watt ME, Reader J, Liebenberg W, Wiesner L, Smith P, Eribez K, Winzeler EA, Kyle DE, Birkholtz LM, Coertzen D, Haynes RK.
Wong HN, et al. Among authors: eribez k.
Front Chem. 2020 Jan 10;7:901. doi: 10.3389/fchem.2019.00901. eCollection 2019.
Front Chem. 2020.
PMID: 31998692
Free PMC article.
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Palstimolide A: A Complex Polyhydroxy Macrolide with Antiparasitic Activity.
Keller L, Siqueira-Neto JL, Souza JM, Eribez K, LaMonte GM, Smith JE, Gerwick WH.
Keller L, et al. Among authors: eribez k.
Molecules. 2020 Mar 31;25(7):1604. doi: 10.3390/molecules25071604.
Molecules. 2020.
PMID: 32244512
Free PMC article.
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Low-latency label-free image-activated cell sorting using fast deep learning and AI inferencing.
Tang R, Xia L, Gutierrez B, Gagne I, Munoz A, Eribez K, Jagnandan N, Chen X, Zhang Z, Waller L, Alaynick W, Cho SH, An C, Lo YH.
Tang R, et al. Among authors: eribez k.
Biosens Bioelectron. 2023 Jan 15;220:114865. doi: 10.1016/j.bios.2022.114865. Epub 2022 Nov 7.
Biosens Bioelectron. 2023.
PMID: 36368140
Free article.
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