Halazy S - Search Results

1

Discovery and development of a new class of potent, selective, orally active oxytocin receptor antagonists.

Quattropani A, Dorbais J, Covini D, Pittet PA, Colovray V, Thomas RJ, Coxhead R, Halazy S, Scheer A, Missotten M, Ayala G, Bradshaw C, De Raemy-Schenk AM, Nichols A, Cirillo R, Tos EG, Giachetti C, Golzio L, Marinelli P, Church DJ, Barberis C, Chollet A, Schwarz MK. Quattropani A, et al. Among authors: halazy s. J Med Chem. 2005 Dec 1;48(24):7882-905. doi: 10.1021/jm050645f. J Med Chem. 2005. PMID: 16302826

2

Design, synthesis, and biological activity of novel, potent, and selective (benzoylaminomethyl)thiophene sulfonamide inhibitors of c-Jun-N-terminal kinase.

Rückle T, Biamonte M, Grippi-Vallotton T, Arkinstall S, Cambet Y, Camps M, Chabert C, Church DJ, Halazy S, Jiang X, Martinou I, Nichols A, Sauer W, Gotteland JP. Rückle T, et al. Among authors: halazy s. J Med Chem. 2004 Dec 30;47(27):6921-34. doi: 10.1021/jm031112e. J Med Chem. 2004. PMID: 15615541

3

Design and synthesis of the first generation of novel potent, selective, and in vivo active (benzothiazol-2-yl)acetonitrile inhibitors of the c-Jun N-terminal kinase.

Gaillard P, Jeanclaude-Etter I, Ardissone V, Arkinstall S, Cambet Y, Camps M, Chabert C, Church D, Cirillo R, Gretener D, Halazy S, Nichols A, Szyndralewiez C, Vitte PA, Gotteland JP. Gaillard P, et al. Among authors: halazy s. J Med Chem. 2005 Jul 14;48(14):4596-607. doi: 10.1021/jm0310986. J Med Chem. 2005. PMID: 15999997

4

Design and synthesis of new potent, silent 5-HT1A antagonists by covalent coupling of aminopropanol derivatives with selective serotonin reuptake inhibitors.

Perez M, Pauwels PJ, Pallard-Sigogneau I, Fourrier C, Chopin P, Palmier C, Colovray V, Halazy S. Perez M, et al. Among authors: halazy s. Bioorg Med Chem Lett. 1998 Dec 1;8(23):3423-8. doi: 10.1016/s0960-894x(98)00619-2. Bioorg Med Chem Lett. 1998. PMID: 9873746

5

In vitro and in vivo pharmacological profile of AS057278, a selective d-amino acid oxidase inhibitor with potential anti-psychotic properties.

Adage T, Trillat AC, Quattropani A, Perrin D, Cavarec L, Shaw J, Guerassimenko O, Giachetti C, Gréco B, Chumakov I, Halazy S, Roach A, Zaratin P. Adage T, et al. Among authors: halazy s. Eur Neuropsychopharmacol. 2008 Mar;18(3):200-14. doi: 10.1016/j.euroneuro.2007.06.006. Epub 2007 Aug 2. Eur Neuropsychopharmacol. 2008. PMID: 17681761

6

3,6-dibromocarbazole piperazine derivatives of 2-propanol as first inhibitors of cytochrome c release via Bax channel modulation.

Bombrun A, Gerber P, Casi G, Terradillos O, Antonsson B, Halazy S. Bombrun A, et al. Among authors: halazy s. J Med Chem. 2003 Oct 9;46(21):4365-8. doi: 10.1021/jm034107j. J Med Chem. 2003. PMID: 14521400

7

Dimerization of sumatriptan as an efficient way to design a potent, centrally and orally active 5-HT1B agonist.

Perez M, Pauwels PJ, Fourrier C, Chopin P, Valentin JP, John GW, Marien M, Halazy S. Perez M, et al. Among authors: halazy s. Bioorg Med Chem Lett. 1998 Mar 17;8(6):675-80. doi: 10.1016/s0960-894x(98)00090-0. Bioorg Med Chem Lett. 1998. PMID: 9871581

8

(Aryloxy)methylsilane derivatives as new cholesterol biosynthesis inhibitors: synthesis and hypocholesterolemic activity of a new class of squalene epoxidase inhibitors.

Gotteland JP, Brunel I, Gendre F, Désiré J, Delhon A, Junquéro D, Oms P, Halazy S. Gotteland JP, et al. Among authors: halazy s. J Med Chem. 1995 Aug 18;38(17):3207-16. doi: 10.1021/jm00017a004. J Med Chem. 1995. PMID: 7650673

9

Serotonin dimers: application of the bivalent ligand approach to the design of new potent and selective 5-HT(1B/1D) agonists.

Halazy S, Perez M, Fourrier C, Pallard I, Pauwels PJ, Palmier C, John GW, Valentin JP, Bonnafous R, Martinez J. Halazy S, et al. J Med Chem. 1996 Dec 6;39(25):4920-7. doi: 10.1021/jm960552l. J Med Chem. 1996. PMID: 8960551

10

Synthesis and serotonergic activity of arylpiperazide derivatives of serotonin: potent agonists for 5-HT1D receptors.

Perez M, Fourrier C, Sigogneau I, Pauwels PJ, Palmier C, John GW, Valentin JP, Halazy S. Perez M, et al. Among authors: halazy s. J Med Chem. 1995 Sep 1;38(18):3602-7. doi: 10.1021/jm00018a020. J Med Chem. 1995. PMID: 7658447

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