Jagdmann GE - Search Results

1

Discovery of N-Substituted 3-Amino-4-(3-boronopropyl)pyrrolidine-3-carboxylic Acids as Highly Potent Third-Generation Inhibitors of Human Arginase I and II.

Van Zandt MC, Jagdmann GE, Whitehouse DL, Ji M, Savoy J, Potapova O, Cousido-Siah A, Mitschler A, Howard EI, Pyle AM, Podjarny AD. Van Zandt MC, et al. Among authors: jagdmann ge. J Med Chem. 2019 Sep 12;62(17):8164-8177. doi: 10.1021/acs.jmedchem.9b00931. Epub 2019 Aug 23. J Med Chem. 2019. PMID: 31408339

2

Discovery of (R)-2-amino-6-borono-2-(2-(piperidin-1-yl)ethyl)hexanoic acid and congeners as highly potent inhibitors of human arginases I and II for treatment of myocardial reperfusion injury.

Van Zandt MC, Whitehouse DL, Golebiowski A, Ji MK, Zhang M, Beckett RP, Jagdmann GE, Ryder TR, Sheeler R, Andreoli M, Conway B, Mahboubi K, D'Angelo G, Mitschler A, Cousido-Siah A, Ruiz FX, Howard EI, Podjarny AD, Schroeter H. Van Zandt MC, et al. Among authors: jagdmann ge. J Med Chem. 2013 Mar 28;56(6):2568-80. doi: 10.1021/jm400014c. Epub 2013 Mar 8. J Med Chem. 2013. PMID: 23472952

3

Small molecules that target group II introns are potent antifungal agents.

Fedorova O, Jagdmann GE Jr, Adams RL, Yuan L, Van Zandt MC, Pyle AM. Fedorova O, et al. Among authors: jagdmann ge jr. Nat Chem Biol. 2018 Dec;14(12):1073-1078. doi: 10.1038/s41589-018-0142-0. Epub 2018 Oct 15. Nat Chem Biol. 2018. PMID: 30323219 Free PMC article.

4

Small-Molecule Antagonists of the RIG-I Innate Immune Receptor.

Rawling DC, Jagdmann GE Jr, Potapova O, Pyle AM. Rawling DC, et al. Among authors: jagdmann ge jr. ACS Chem Biol. 2020 Feb 21;15(2):311-317. doi: 10.1021/acschembio.9b00810. Epub 2020 Jan 27. ACS Chem Biol. 2020. PMID: 31944652

5

Chemical synthesis and characterization of epicatechin glucuronides and sulfates: bioanalytical standards for epicatechin metabolite identification.

Zhang M, Jagdmann GE Jr, Van Zandt M, Sheeler R, Beckett P, Schroeter H. Zhang M, et al. Among authors: jagdmann ge jr. J Nat Prod. 2013 Feb 22;76(2):157-69. doi: 10.1021/np300568m. Epub 2013 Jan 28. J Nat Prod. 2013. PMID: 23356946 Free article.

6

Synthesis and protein kinase inhibitory activity of balanol analogues with modified benzophenone subunits.

Lampe JW, Biggers CK, Defauw JM, Foglesong RJ, Hall SE, Heerding JM, Hollinshead SP, Hu H, Hughes PF, Jagdmann GE Jr, Johnson MG, Lai YS, Lowden CT, Lynch MP, Mendoza JS, Murphy MM, Wilson JW, Ballas LM, Carter K, Darges JW, Davis JE, Hubbard FR, Stamper ML. Lampe JW, et al. Among authors: jagdmann ge jr. J Med Chem. 2002 Jun 6;45(12):2624-43. doi: 10.1021/jm020018f. J Med Chem. 2002. PMID: 12036372

7

Discovery of allosteric potentiators for the metabotropic glutamate 2 receptor: synthesis and subtype selectivity of N-(4-(2-methoxyphenoxy)phenyl)-N-(2,2,2- trifluoroethylsulfonyl)pyrid-3-ylmethylamine.

Johnson MP, Baez M, Jagdmann GE Jr, Britton TC, Large TH, Callagaro DO, Tizzano JP, Monn JA, Schoepp DD. Johnson MP, et al. Among authors: jagdmann ge jr. J Med Chem. 2003 Jul 17;46(15):3189-92. doi: 10.1021/jm034015u. J Med Chem. 2003. PMID: 12852748

8

SAR study of a subtype selective allosteric potentiator of metabotropic glutamate 2 receptor, N-(4-phenoxyphenyl)-N-(3-pyridinylmethyl)ethanesulfonamide.

Barda DA, Wang ZQ, Britton TC, Henry SS, Jagdmann GE, Coleman DS, Johnson MP, Andis SL, Schoepp DD. Barda DA, et al. Among authors: jagdmann ge. Bioorg Med Chem Lett. 2004 Jun 21;14(12):3099-102. doi: 10.1016/j.bmcl.2004.04.017. Bioorg Med Chem Lett. 2004. PMID: 15149652

9

Synthesis and protein kinase C inhibitory activities of acyclic balanol analogs that are highly selective for protein kinase C over protein kinase A.

Defauw JM, Murphy MM, Jagdmann GE Jr, Hu H, Lampe JW, Hollinshead SP, Mitchell TJ, Crane HM, Heerding JM, Mendoza JS, Davis JE, Darges JW, Hubbard FR, Hall SE. Defauw JM, et al. Among authors: jagdmann ge jr. J Med Chem. 1996 Dec 20;39(26):5215-27. doi: 10.1021/jm960581w. J Med Chem. 1996. PMID: 8978850

10

Synthesis and protein kinase C inhibitory activities of balanol analogs with replacement of the perhydroazepine moiety.

Lai YS, Mendoza JS, Jagdmann GE Jr, Menaldino DS, Biggers CK, Heerding JM, Wilson JW, Hall SE, Jiang JB, Janzen WP, Ballas LM. Lai YS, et al. Among authors: jagdmann ge jr. J Med Chem. 1997 Jan 17;40(2):226-35. doi: 10.1021/jm960497g. J Med Chem. 1997. PMID: 9003521

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