Klotz KN - Search Results

1

Combining selectivity and affinity predictions using an integrated Support Vector Machine (SVM) approach: An alternative tool to discriminate between the human adenosine A(2A) and A(3) receptor pyrazolo-triazolo-pyrimidine antagonists binding sites.

Michielan L, Bolcato C, Federico S, Cacciari B, Bacilieri M, Klotz KN, Kachler S, Pastorin G, Cardin R, Sperduti A, Spalluto G, Moro S. Michielan L, et al. Among authors: klotz kn. Bioorg Med Chem. 2009 Jul 15;17(14):5259-74. doi: 10.1016/j.bmc.2009.05.038. Epub 2009 May 21. Bioorg Med Chem. 2009. PMID: 19501513

2

2-Alkynyl derivatives of adenosine and adenosine-5'-N-ethyluronamide as selective agonists at A2 adenosine receptors.

Cristalli G, Eleuteri A, Vittori S, Volpini R, Lohse MJ, Klotz KN. Cristalli G, et al. Among authors: klotz kn. J Med Chem. 1992 Jun 26;35(13):2363-8. doi: 10.1021/jm00091a003. J Med Chem. 1992. PMID: 1619615

3

Adenosine receptor agonists: synthesis and biological evaluation of 1-deaza analogues of adenosine derivatives.

Cristalli G, Franchetti P, Grifantini M, Vittori S, Klotz KN, Lohse MJ. Cristalli G, et al. Among authors: klotz kn. J Med Chem. 1988 Jun;31(6):1179-83. doi: 10.1021/jm00401a018. J Med Chem. 1988. PMID: 3373486

4

Synthesis of new delta 2-isoxazoline derivatives and their pharmacological characterization as beta-adrenergic receptor antagonists.

Conti P, Dallanoce C, De Amici M, De Micheli C, Klotz KN. Conti P, et al. Among authors: klotz kn. Bioorg Med Chem. 1998 Apr;6(4):401-8. doi: 10.1016/s0968-0896(97)10051-7. Bioorg Med Chem. 1998. PMID: 9597184

5

New substituted 9-alkylpurines as adenosine receptor ligands.

Camaioni E, Costanzi S, Vittori S, Volpini R, Klotz KN, Cristalli G. Camaioni E, et al. Among authors: klotz kn. Bioorg Med Chem. 1998 May;6(5):523-33. doi: 10.1016/s0968-0896(98)00007-8. Bioorg Med Chem. 1998. PMID: 9629466

6

8-(Sulfostyryl)xanthines: water-soluble A2A-selective adenosine receptor antagonists.

Müller CE, Sandoval-Ramírez J, Schobert U, Geis U, Frobenius W, Klotz KN. Müller CE, et al. Among authors: klotz kn. Bioorg Med Chem. 1998 Jun;6(6):707-19. doi: 10.1016/s0968-0896(98)00025-x. Bioorg Med Chem. 1998. PMID: 9681137

7

Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives as highly potent and selective human A(3) adenosine receptor antagonists.

Baraldi PG, Cacciari B, Romagnoli R, Spalluto G, Klotz KN, Leung E, Varani K, Gessi S, Merighi S, Borea PA. Baraldi PG, et al. Among authors: klotz kn. J Med Chem. 1999 Nov 4;42(22):4473-8. doi: 10.1021/jm991114s. J Med Chem. 1999. PMID: 10579811 No abstract available.

8

Synthesis of di- and tri-substituted adenosine derivatives and their affinities at human adenosine receptor subtypes.

Volpini R, Camaioni E, Costanzi S, Vittori S, Klotz KN, Cristalli G. Volpini R, et al. Among authors: klotz kn. Nucleosides Nucleotides. 1999 Nov-Dec;18(11-12):2511-20. doi: 10.1080/07328319908044623. Nucleosides Nucleotides. 1999. PMID: 10639752

9

[(3)H]MRE 3008F20: a novel antagonist radioligand for the pharmacological and biochemical characterization of human A(3) adenosine receptors.

Varani K, Merighi S, Gessi S, Klotz KN, Leung E, Baraldi PG, Cacciari B, Romagnoli R, Spalluto G, Borea PA. Varani K, et al. Among authors: klotz kn. Mol Pharmacol. 2000 May;57(5):968-75. Mol Pharmacol. 2000. PMID: 10779381

10

7-Deazaadenines bearing polar substituents: structure-activity relationships of new A(1) and A(3) adenosine receptor antagonists.

Hess S, Müller CE, Frobenius W, Reith U, Klotz KN, Eger K. Hess S, et al. Among authors: klotz kn. J Med Chem. 2000 Nov 30;43(24):4636-46. doi: 10.1021/jm000967d. J Med Chem. 2000. PMID: 11101355

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