Korfmacher WA - Search Results

1

Novel procedure for rapid pharmacokinetic screening of discovery compounds in rats.

Cox KA, Dunn-Meynell K, Korfmacher WA, Broske L, Nomeir AA, Lin CC, Cayen MN, Barr WH. Cox KA, et al. Among authors: korfmacher wa. Drug Discov Today. 1999 May;4(5):232-237. doi: 10.1016/s1359-6446(98)01299-9. Drug Discov Today. 1999. PMID: 10322290

2

Characterization of the nociceptin receptor (ORL-1) agonist, Ro64-6198, in tests of anxiety across multiple species.

Varty GB, Hyde LA, Hodgson RA, Lu SX, McCool MF, Kazdoba TM, Del Vecchio RA, Guthrie DH, Pond AJ, Grzelak ME, Xu X, Korfmacher WA, Tulshian D, Parker EM, Higgins GA. Varty GB, et al. Among authors: korfmacher wa. Psychopharmacology (Berl). 2005 Oct;182(1):132-43. doi: 10.1007/s00213-005-0041-4. Epub 2005 Sep 29. Psychopharmacology (Berl). 2005. PMID: 16025321

3

Synthesis and SAR studies of benzimidazolone derivatives as histamine H3-receptor antagonists.

Zeng Q, Rosenblum SB, Yang Z, Jiang Y, McCormick KD, Aslanian RG, Duguma L, Kozlowski JA, Shih NY, Hey JA, West RE Jr, Korfmacher WA, Berlin M, Boyce CW. Zeng Q, et al. Among authors: korfmacher wa. Bioorg Med Chem Lett. 2013 Nov 1;23(21):6001-3. doi: 10.1016/j.bmcl.2013.08.012. Epub 2013 Aug 13. Bioorg Med Chem Lett. 2013. PMID: 24050887

4

Fused bicycles as arylketone bioisosteres leading to potent, orally active thiadiazole H3 antagonists.

Xiao D, Palani A, Sofolarides M, Aslanian R, West RE Jr, Williams SM, Wu RL, Hwa J, Sondey C, Lachowicz J, Korfmacher WA. Xiao D, et al. Among authors: korfmacher wa. Bioorg Med Chem Lett. 2012 May 1;22(9):3354-7. doi: 10.1016/j.bmcl.2012.02.076. Epub 2012 Mar 8. Bioorg Med Chem Lett. 2012. PMID: 22464130

5

Liquid extraction surface analysis mass spectrometry (LESA-MS) as a novel profiling tool for drug distribution and metabolism analysis: the terfenadine example.

Eikel D, Vavrek M, Smith S, Bason C, Yeh S, Korfmacher WA, Henion JD. Eikel D, et al. Among authors: korfmacher wa. Rapid Commun Mass Spectrom. 2011 Dec 15;25(23):3587-96. doi: 10.1002/rcm.5274. Rapid Commun Mass Spectrom. 2011. PMID: 22095508

6

It is time for a paradigm shift in drug discovery bioanalysis: from SRM to HRMS.

Ramanathan R, Jemal M, Ramagiri S, Xia YQ, Humpreys WG, Olah T, Korfmacher WA. Ramanathan R, et al. Among authors: korfmacher wa. J Mass Spectrom. 2011 Jun;46(6):595-601. doi: 10.1002/jms.1921. J Mass Spectrom. 2011. PMID: 21630388

7

The synthesis and structure-activity relationship of 4-benzimidazolyl-piperidinylcarbonyl-piperidine analogs as histamine H3 antagonists.

Ting PC, Lee JF, Albanese MM, Wu J, Aslanian R, Favreau L, Nardo C, Korfmacher WA, West RE, Williams SM, Anthes JC, Rivelli MA, Corboz MR, Hey JA. Ting PC, et al. Among authors: korfmacher wa. Bioorg Med Chem Lett. 2010 Sep 1;20(17):5004-8. doi: 10.1016/j.bmcl.2010.07.052. Epub 2010 Jul 16. Bioorg Med Chem Lett. 2010. PMID: 20685118

8

Mapping pharmaceuticals in rat brain sections using MALDI imaging mass spectrometry.

Hsieh Y, Li F, Korfmacher WA. Hsieh Y, et al. Among authors: korfmacher wa. Methods Mol Biol. 2010;656:147-58. doi: 10.1007/978-1-60761-746-4_8. Methods Mol Biol. 2010. PMID: 20680589

9

The role of exploratory drug metabolism and pharmacokinetics in new drug research: case study-selection of a thrombin receptor antagonist for development.

Hsieh Y, Cheng KC, Wang Y, Chackalamannil S, Xia Y, Korfmacher WA, White RE. Hsieh Y, et al. Among authors: korfmacher wa. Curr Pharm Des. 2009;15(19):2262-9. doi: 10.2174/138161209788682497. Curr Pharm Des. 2009. PMID: 19601827

10

Advances in the integration of drug metabolism into the lead optimization paradigm.

Korfmacher WA. Korfmacher WA. Mini Rev Med Chem. 2009 Jun;9(6):703-16. doi: 10.2174/138955709788452694. Mini Rev Med Chem. 2009. PMID: 19519496 Review.

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