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Genome-Wide CRISPR Screen for Essential Cell Growth Mediators in Mutant KRAS Colorectal Cancers.
Cancer Res. 2017 Nov 15;77(22):6330-6339. doi: 10.1158/0008-5472.CAN-17-2043. Epub 2017 Sep 27.
Cancer Res. 2017.
PMID: 28954733
Free PMC article.
1,2,3-Triazoles as Amide Bioisosteres: Discovery of a New Class of Potent HIV-1 Vif Antagonists.
Mohammed I, Kummetha IR, Singh G, Sharova N, Lichinchi G, Dang J, Stevenson M, Rana TM.
Mohammed I, et al. Among authors: kummetha ir.
J Med Chem. 2016 Aug 25;59(16):7677-82. doi: 10.1021/acs.jmedchem.6b00247. Epub 2016 Aug 10.
J Med Chem. 2016.
PMID: 27509004
Free PMC article.
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HIV-1 Escape from Small-Molecule Antagonism of Vif.
Sharkey M, Sharova N, Mohammed I, Huff SE, Kummetha IR, Singh G, Rana TM, Stevenson M.
Sharkey M, et al. Among authors: kummetha ir.
mBio. 2019 Feb 26;10(1):e00144-19. doi: 10.1128/mBio.00144-19.
mBio. 2019.
PMID: 30808702
Free PMC article.
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Discovery and Mechanism of SARS-CoV-2 Main Protease Inhibitors.
Huff S, Kummetha IR, Tiwari SK, Huante MB, Clark AE, Wang S, Bray W, Smith D, Carlin AF, Endsley M, Rana TM.
Huff S, et al. Among authors: kummetha ir.
J Med Chem. 2022 Feb 24;65(4):2866-2879. doi: 10.1021/acs.jmedchem.1c00566. Epub 2021 Sep 27.
J Med Chem. 2022.
PMID: 34570513
Free PMC article.
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Rational Design and Optimization of m6A-RNA Demethylase FTO Inhibitors as Anticancer Agents.
Huff S, Kummetha IR, Zhang L, Wang L, Bray W, Yin J, Kelley V, Wang Y, Rana TM.
Huff S, et al. Among authors: kummetha ir.
J Med Chem. 2022 Aug 25;65(16):10920-10937. doi: 10.1021/acs.jmedchem.1c02075. Epub 2022 Aug 8.
J Med Chem. 2022.
PMID: 35939803
Free PMC article.
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Small-molecule PTPN2 Inhibitors Sensitize Resistant Melanoma to Anti-PD-1 Immunotherapy.
Zhu Z, Tang R, Huff S, Kummetha IR, Wang L, Li N, Rana TM.
Zhu Z, et al. Among authors: kummetha ir.
Cancer Res Commun. 2023 Jan 24;3(1):119-129. doi: 10.1158/2767-9764.CRC-21-0186. eCollection 2023 Jan.
Cancer Res Commun. 2023.
PMID: 36968224
Free PMC article.
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