Leung E - Search Results

1

Synthesis and biological effects of a new series of 2-amino-3-benzoylthiophenes as allosteric enhancers of A1-adenosine receptor.

Baraldi PG, Zaid AN, Lampronti I, Fruttarolo F, Pavani MG, Tabrizi MA, Shryock JC, Leung E, Romagnoli R. Baraldi PG, et al. Among authors: leung e. Bioorg Med Chem Lett. 2000 Sep 4;10(17):1953-7. doi: 10.1016/s0960-894x(00)00379-6. Bioorg Med Chem Lett. 2000. PMID: 10987425

2

Synthesis and biological effects of novel 2-amino-3-naphthoylthiophenes as allosteric enhancers of the A1 adenosine receptor.

Baraldi PG, Romagnoli R, Pavani MG, Nuñez Mdel C, Tabrizi MA, Shryock JC, Leung E, Moorman AR, Uluoglu C, Iannotta V, Merighi S, Borea PA. Baraldi PG, et al. Among authors: leung e. J Med Chem. 2003 Feb 27;46(5):794-809. doi: 10.1021/jm0210212. J Med Chem. 2003. PMID: 12593659

3

Synthesis and biological characterization of [3H] (2-amino-4,5,6,7-tetrahydrobenzo[b]thiophen-3-yl)-(4-chlorophenyl)-methanone, the first radiolabelled adenosine A1 allosteric enhancer.

Baraldi PG, Pavani MG, Leung E, Moorman AR, Varani K, Vincenzi F, Borea PA, Romagnoli R. Baraldi PG, et al. Among authors: leung e. Bioorg Med Chem Lett. 2006 Mar 1;16(5):1402-4. doi: 10.1016/j.bmcl.2005.11.037. Bioorg Med Chem Lett. 2006. PMID: 16321527

4

Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives as highly potent and selective human A(3) adenosine receptor antagonists: influence of the chain at the N(8) pyrazole nitrogen.

Baraldi PG, Cacciari B, Romagnoli R, Spalluto G, Moro S, Klotz KN, Leung E, Varani K, Gessi S, Merighi S, Borea PA. Baraldi PG, et al. Among authors: leung e. J Med Chem. 2000 Dec 14;43(25):4768-80. doi: 10.1021/jm001047y. J Med Chem. 2000. PMID: 11123985

5

Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives as highly potent and selective human A(3) adenosine receptor antagonists.

Baraldi PG, Cacciari B, Romagnoli R, Spalluto G, Klotz KN, Leung E, Varani K, Gessi S, Merighi S, Borea PA. Baraldi PG, et al. Among authors: leung e. J Med Chem. 1999 Nov 4;42(22):4473-8. doi: 10.1021/jm991114s. J Med Chem. 1999. PMID: 10579811 No abstract available.

6

Synthesis and preliminary biological evaluation of [3H]-MRE 3008-F20: the first high affinity radioligand antagonist for the human A3 adenosine receptors.

Baraldi PG, Cacciari B, Romagnoli R, Varani K, Merighi S, Gessi S, Borea PA, Leung E, Hickey SL, Spalluto G. Baraldi PG, et al. Among authors: leung e. Bioorg Med Chem Lett. 2000 Feb 7;10(3):209-11. doi: 10.1016/s0960-894x(99)00674-5. Bioorg Med Chem Lett. 2000. PMID: 10698437

7

[(3)H]MRE 3008F20: a novel antagonist radioligand for the pharmacological and biochemical characterization of human A(3) adenosine receptors.

Varani K, Merighi S, Gessi S, Klotz KN, Leung E, Baraldi PG, Cacciari B, Romagnoli R, Spalluto G, Borea PA. Varani K, et al. Among authors: leung e. Mol Pharmacol. 2000 May;57(5):968-75. Mol Pharmacol. 2000. PMID: 10779381

8

Pharmacological and biochemical characterization of A3 adenosine receptors in Jurkat T cells.

Gessi S, Varani K, Merighi S, Morelli A, Ferrari D, Leung E, Baraldi PG, Spalluto G, Borea PA. Gessi S, et al. Among authors: leung e. Br J Pharmacol. 2001 Sep;134(1):116-26. doi: 10.1038/sj.bjp.0704254. Br J Pharmacol. 2001. PMID: 11522603 Free PMC article.

9

Binding thermodynamics at the human A(3) adenosine receptor.

Merighi S, Varani K, Gessi S, Klotz KN, Leung E, Baraldi PG, Borea PA. Merighi S, et al. Among authors: leung e. Biochem Pharmacol. 2002 Jan 15;63(2):157-61. doi: 10.1016/s0006-2952(01)00825-5. Biochem Pharmacol. 2002. PMID: 11841789

10

A glance at adenosine receptors: novel target for antitumor therapy.

Merighi S, Mirandola P, Varani K, Gessi S, Leung E, Baraldi PG, Tabrizi MA, Borea PA. Merighi S, et al. Among authors: leung e. Pharmacol Ther. 2003 Oct;100(1):31-48. doi: 10.1016/s0163-7258(03)00084-6. Pharmacol Ther. 2003. PMID: 14550503 Review.

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