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THC shows activity against cultured Plasmodium falciparum.
Bioorg Med Chem Lett. 2021 Dec 15;54:128442. doi: 10.1016/j.bmcl.2021.128442. Epub 2021 Nov 8.
Bioorg Med Chem Lett. 2021.
PMID: 34763083
Identification of 2,4-Disubstituted Imidazopyridines as Hemozoin Formation Inhibitors with Fast-Killing Kinetics and In Vivo Efficacy in the Plasmodium falciparum NSG Mouse Model.
Horatscheck A, Andrijevic A, Nchinda AT, Le Manach C, Paquet T, Khonde LP, Dam J, Pawar K, Taylor D, Lawrence N, Brunschwig C, Gibhard L, Njoroge M, Reader J, van der Watt M, Wicht K, de Sousa ACC, Okombo J, Maepa K, Egan TJ, Birkholtz LM, Basarab GS, Wittlin S, Fish PV, Street LJ, Duffy J, Chibale K.
Horatscheck A, et al. Among authors: maepa k.
J Med Chem. 2020 Nov 12;63(21):13013-13030. doi: 10.1021/acs.jmedchem.0c01411. Epub 2020 Oct 25.
J Med Chem. 2020.
PMID: 33103428
Free PMC article.
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A Diverse Range of Hemozoin Inhibiting Scaffolds Act on Plasmodium falciparum as Heme Complexes.
Openshaw R, Maepa K, Benjamin SJ, Wainwright L, Combrinck JM, Hunter R, Egan TJ.
Openshaw R, et al. Among authors: maepa k.
ACS Infect Dis. 2021 Feb 12;7(2):362-376. doi: 10.1021/acsinfecdis.0c00680. Epub 2021 Jan 12.
ACS Infect Dis. 2021.
PMID: 33430579
Free PMC article.
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Virtual screening as a tool to discover new β-haematin inhibitors with activity against malaria parasites.
de Sousa ACC, Combrinck JM, Maepa K, Egan TJ.
de Sousa ACC, et al. Among authors: maepa k.
Sci Rep. 2020 Feb 25;10(1):3374. doi: 10.1038/s41598-020-60221-0.
Sci Rep. 2020.
PMID: 32099045
Free PMC article.
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Lapatinib, Nilotinib and Lomitapide Inhibit Haemozoin Formation in Malaria Parasites.
de Sousa ACC, Maepa K, Combrinck JM, Egan TJ.
de Sousa ACC, et al. Among authors: maepa k.
Molecules. 2020 Mar 29;25(7):1571. doi: 10.3390/molecules25071571.
Molecules. 2020.
PMID: 32235391
Free PMC article.
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Correction to "Identification of 2,4-Disubstituted Imidazopyridines as Hemozoin Formation Inhibitors with Fast-Killing Kinetics and In Vivo Efficacy in the Plasmodium falciparum NSG Mouse Model".
Horatscheck A, Andrijevic A, Nchinda AT, Le Manach C, Paquet T, Khonde LP, Dam J, Pawar K, Taylor D, Lawrence N, Brunschwig C, Gibhard L, Njoroge M, Reader J, van der Watt M, Wicht K, de Sousa ACC, Okombo J, Maepa K, Egan TJ, Birkholtz LM, Basarab GS, Wittlin S, Fish PV, Street LJ, Duffy J, Chibale K.
Horatscheck A, et al. Among authors: maepa k.
J Med Chem. 2021 Feb 11;64(3):1762. doi: 10.1021/acs.jmedchem.1c00064. Epub 2021 Jan 28.
J Med Chem. 2021.
PMID: 33508187
No abstract available.
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Structure-activity relationship studies of antiplasmodial cyclometallated ruthenium(II), rhodium(III) and iridium(III) complexes of 2-phenylbenzimidazoles.
Rylands LI, Welsh A, Maepa K, Stringer T, Taylor D, Chibale K, Smith GS.
Rylands LI, et al. Among authors: maepa k.
Eur J Med Chem. 2019 Jan 1;161:11-21. doi: 10.1016/j.ejmech.2018.10.019. Epub 2018 Oct 10.
Eur J Med Chem. 2019.
PMID: 30342422
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