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Page 1
VHL-Modified PROteolysis TArgeting Chimeras (PROTACs) as a Strategy to Evade Metabolic Degradation in In Vitro Applications.
J Med Chem. 2023 Sep 28;66(18):13148-13171. doi: 10.1021/acs.jmedchem.3c01144. Epub 2023 Sep 12.
J Med Chem. 2023.
PMID: 37699425
PROTACs bearing piperazine-containing linkers: what effect on their protonation state?
Desantis J, Mammoli A, Eleuteri M, Coletti A, Croci F, Macchiarulo A, Goracci L.
Desantis J, et al. Among authors: eleuteri m.
RSC Adv. 2022 Aug 9;12(34):21968-21977. doi: 10.1039/d2ra03761k. eCollection 2022 Aug 4.
RSC Adv. 2022.
PMID: 36043064
Free PMC article.
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Discovery of novel SARS-CoV-2 inhibitors targeting the main protease Mpro by virtual screenings and hit optimization.
Mercorelli B, Desantis J, Celegato M, Bazzacco A, Siragusa L, Benedetti P, Eleuteri M, Croci F, Cruciani G, Goracci L, Loregian A.
Mercorelli B, et al. Among authors: eleuteri m.
Antiviral Res. 2022 Aug;204:105350. doi: 10.1016/j.antiviral.2022.105350. Epub 2022 Jun 7.
Antiviral Res. 2022.
PMID: 35688349
Free PMC article.
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Understanding the Metabolism of Proteolysis Targeting Chimeras (PROTACs): The Next Step toward Pharmaceutical Applications.
Goracci L, Desantis J, Valeri A, Castellani B, Eleuteri M, Cruciani G.
Goracci L, et al. Among authors: eleuteri m.
J Med Chem. 2020 Oct 22;63(20):11615-11638. doi: 10.1021/acs.jmedchem.0c00793. Epub 2020 Oct 7.
J Med Chem. 2020.
PMID: 33026811
Free PMC article.
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Use of ionic liquids in amidation reactions for proteolysis targeting chimera synthesis.
Eleuteri M, Desantis J, Cruciani G, Germani R, Goracci L.
Eleuteri M, et al.
Org Biomol Chem. 2024 Apr 11. doi: 10.1039/d4ob00304g. Online ahead of print.
Org Biomol Chem. 2024.
PMID: 38602033
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Design, synthesis, and biological evaluation of first-in-class indomethacin-based PROTACs degrading SARS-CoV-2 main protease and with broad-spectrum antiviral activity.
Desantis J, Bazzacco A, Eleuteri M, Tuci S, Bianconi E, Macchiarulo A, Mercorelli B, Loregian A, Goracci L.
Desantis J, et al. Among authors: eleuteri m.
Eur J Med Chem. 2024 Mar 15;268:116202. doi: 10.1016/j.ejmech.2024.116202. Epub 2024 Feb 6.
Eur J Med Chem. 2024.
PMID: 38394929
Free article.
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